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1-(2,3,5,6-tetramethylbenzoyl)azetidin-3-ol
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-(carbamoylmethyl)-N-(3-hydroxyadamantan-1-yl)piperidine-3-carboxamide
N-(2-hydroxyethyl)-3-(4-methyl-1,3-thiazol-5-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
1-{[4-(methylsulfanyl)phenyl]methyl}-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
8-[(2,3-dimethoxyphenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(4-aminoazepan-1-yl)-3-oxopropyl]-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
2-methoxy-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
9-[(5-chloro-2-fluorophenyl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
1-(1-cyclobutylpiperidin-3-yl)-4-(2-fluorophenyl)piperazine
5-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(2-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
1-[(4-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
(1R,3S)-7-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-7-azaspiro[3.5]nonane-1,3-diol
2-methyl-4-(2-methylphenyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
1-{2-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]pyrimidin-4-yl}pyrrolidin-3-ol
[3-(2-methoxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]methanol
2-({[(3R,4R)-1-[(2,4-dichlorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
propan-2-yl 2-chloro-5-{[methyl(1,2-oxazol-3-ylmethyl)carbamoyl]amino}benzoate
3-(2-methyl-1-benzofuran-7-yl)-1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]urea
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(3-methylphenoxy)azetidine
3-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-4,6-dimethylpyrimidine
methyl (2S)-2-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]amino}propanoate
(3S,4S)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-[2-(3-methylbutoxy)phenyl]-1H-imidazole
3-(piperidine-1-carbonyl)-N-(thiolan-3-yl)pyrazine-2-carboxamide
(2R,3R)-1'-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-cyclopentyl-5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]piperidin-2-one
methyl 5-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
[2-({1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperidin-4-yl}oxy)ethyl]dimethylamine
2-{[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
2-[(1-benzylpyrrolidin-3-yl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(butan-2-yl)-N-[(3-methylthiophen-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(1-{[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
4-methoxy-6-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
3-({1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
8-(2-hydroxy-3-methylbutanoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(dicyclopropylmethyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-{1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(methylsulfanyl)pyrimidine-5-carboxylate
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3-dimethoxybenzamide
1-methyl-2-(morpholin-4-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-amino-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
N3-butyl-1-(furan-2-ylmethyl)-4-oxo-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
[2-methoxy-5-(1H-pyrazol-3-yl)phenyl]methanol
2-(pyridin-3-yl)-N-[1-(thiophen-2-yl)propyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)phenol