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2-methyl-5-[3-(2-propyl-1H-imidazol-1-yl)phenyl]-1,3,4-thiadiazole
1-(2-{2,8-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
(butan-2-yl)[(1-ethyl-1H-pyrazol-4-yl)methyl](3-phenylprop-2-yn-1-yl)amine
2,3-difluoro-6-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
1'-(1,4-dithiepan-6-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 2-(diethylsulfamoyl)-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 2-({5-[({2-[(prop-2-en-1-yl)amino]phenyl}formamido)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)acetate
N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]acetamide
(3R,4R)-4-ethyl-1-[2-methyl-5-(trifluoromethyl)benzoyl]piperidine-3,4-diol
(3S,9aR)-8-(4-phenylbenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-imidazol-1-yl)propyl]amine
4-(benzyloxy)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(oxolan-2-ylmethyl)amino]pyridine-3-carboxamide
3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-(dimethyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2,3-dihydro-1H-inden-2-amine
N-(2-{4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenoxy}ethyl)acetamide
N,3,5,7-tetramethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
[4-({1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)quinazolin-2-yl]methanol
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
(1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
4-{[2-(2-fluorophenyl)ethyl]amino}-N-(2-hydroxy-2-phenylethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-(benzyloxy)-1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-[(2,3-difluorophenyl)methyl]-3-({[(5,6-dimethylpyridin-3-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-methyl-2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)acetamide
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[1-(methoxymethyl)cyclopentyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(2-fluorophenyl)methyl]-1,4-diazepane
2-[2-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-[(2-ethoxypyridin-3-yl)methyl]-2-ethylpyrimidine-5-carboxamide
2-(3-fluoro-2,4-dimethylphenyl)-1-(3-methoxypropyl)-1H-imidazole
4-chloro-N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-2-(thiophen-2-yl)pyrimidine
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
7-[2-(3-methoxyphenoxy)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-4-methoxy-2-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(4-methyl-1,3-oxazole-5-carbonyl)-decahydro-1,6-naphthyridine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-fluorophenyl)ethyl]acetamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
8-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-oxa-8-azaspiro[4.5]decane
5-(5-chlorothiophen-2-yl)pyridine-3-carboxylic acid
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-(3-hydroxypropyl)-1-methyl-N-(thiophen-2-ylmethyl)-1H-indole-4-carboxamide
N,N-dimethyl-2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine-3-carboxamide
4-ethyl-5-methyl-N-{2-[methyl(phenyl)amino]propyl}pyrimidin-2-amine
N-({1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)furan-2-carboxamide