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2-(morpholin-4-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
1-{2-[4-(dimethylamino)azepan-1-yl]-2-oxoethyl}-2-methyl-1H-indole-3-carbonitrile
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-5-propyl-1,2-oxazole
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
6,7-dimethoxy-2-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
2,4-dimethyl-5-({2-[(pyridin-3-yl)amino]ethyl}carbamoyl)-1H-pyrrole-3-carboxylic acid
N-[(3R,4S)-1-cyclohexyl-4-cyclopropylpyrrolidin-3-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2,2-diphenylethan-1-one
6-{4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-cyclohexyl-1,4-diazepane
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}[(1-ethylpiperidin-3-yl)methyl]methylamine
4-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-{4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxymethyl}pyridine
3-(2-chlorophenyl)-1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine
1-methyl-3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinoxalin-2-one
prop-2-en-1-yl 3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
(3S,4R)-4-methyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidine-3,4-diol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}furan-2-carboxamide
N-[(2R,4R,6S)-2-tert-butyl-6-(2-butyl-5-chloro-1H-imidazol-4-yl)oxan-4-yl]acetamide
dimethyl({3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl})amine
4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
N-methyl-N-(pyridin-2-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-(2-methoxyethyl)-1-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
2-amino-8-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-(2,3-difluorophenoxymethyl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
1-(1H-indazol-6-yl)-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazin-2-one
N-[3-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}[1-(2-fluorophenyl)propan-2-yl]amine
N-{4-[3-(ethanesulfinyl)propanamido]phenyl}-5-methylfuran-2-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
1-(2-phenylethyl)-4-[4-(propan-2-yl)pyrimidin-2-yl]piperazin-2-one
1-[4-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-one
2-(5-acetylthiophen-3-yl)-1-{4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
(4aR,7aS)-1-(2-methylpropyl)-4-[2-(6-methylpyridin-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(5-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-2-[3-(pyridin-3-yl)-1H-indazol-1-yl]acetamide
(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-[(thiophen-3-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3S,5R)-N-(6-methylpyridin-3-yl)-5-(thiomorpholine-4-carbonyl)piperidine-3-carboxamide
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidine
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
2,3-dimethyl-N-[3-(methylsulfamoyl)phenyl]-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
6-(3,4,5-trimethoxyphenyl)-1H-indole
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide