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1-(furan-3-ylmethyl)-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-[(3-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(furan-2-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-phenylpropanamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(4,4,4-trifluorobutyl)piperidin-3-yl]propanamide
2-methyl-3-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]propanoic acid
N-(furan-2-ylmethyl)-2-methanesulfonyl-N-[2-(morpholin-4-yl)ethyl]acetamide
5-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-1H-indole
1-({1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-(3-methylphenyl)ethan-1-one
3-(cyclopropylsulfamoyl)-5-(3,4,5-trifluorophenyl)benzoic acid
2-(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
2-(1-methyl-1H-imidazol-2-yl)-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
3-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
2-(ethylamino)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrimidine-5-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
(1S,5R)-3-(1H-1,3-benzodiazol-2-ylmethyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-[3-(1H-pyrazol-1-yl)phenyl]urea
5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-methyl-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-1-propyl-1H-pyrazole-4-carboxamide
1-{[2-(5-chloro-2-methoxyphenyl)phenyl]methyl}piperazine
N-(1,3-benzoxazol-2-ylmethyl)-1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
(4aR,7aS)-1-propyl-4-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2H-indazol-2-yl)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(1H-pyrazol-1-yl)benzamide
3-butyl-4-ethyl-1-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-4,6-dimethylpyrimidin-2-amine
3-ethyl-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-cyclohexyl-5-[(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)methyl]pyrimidine
1-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({5-cyclopentyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)methylamine
6-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,3-benzothiazole
(1S,5R)-6-(naphthalen-2-ylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-fluorophenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-({7-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1,3-thiazole
5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
6-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-phenylpropanamide
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-(3-fluorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carbonyl]piperazin-2-one
methyl 4-({2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}methyl)benzoate
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]urea
3-(4-methoxyphenyl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide