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2-(3-fluoro-4-methoxyphenyl)-5,6-dimethylpyridine-3-carboxamide
8-methoxy-N-methyl-N-(1,2-oxazol-5-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aS,7aR)-1-(3-chloro-5-fluorobenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-cycloheptyl-N-ethyl-1,2-oxazole-3-carboxamide
1-(4-fluorophenyl)-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]benzamide
2-methyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
6-{[2-(1H-imidazol-4-yl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-ethyl-9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-phenyl-2,9-diazaspiro[5.5]undecane
3-chloro-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-methoxy-N-methylbenzamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-hydroxy-3-methylbutan-2-yl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-chloro-4-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-4-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-benzyl-N-methyl-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1H-1,2,3-triazol-4-ylmethyl)piperidin-4-ol
1-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-4-phenylpyrrolidin-2-one
N-[(3R,4S)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-[(3R,4R)-3-hydroxy-1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
4-[4-(4-methoxyphenoxy)piperidin-1-yl]-5,6-dimethylpyrimidine
[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-(1-methyl-1H-indazol-3-yl)-2-[3-(3-methylquinoxalin-2-yl)-1H-pyrazol-1-yl]acetamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
(furan-2-ylmethyl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})(3-methylbutan-2-yl)amine
[(2,2-dimethyloxan-4-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-methyl-2-({[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
2-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
8-methoxy-N-[2-(3-methylpyridin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
1-(isoquinoline-5-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
2-[4-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperazin-1-yl]benzonitrile
6-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
1-(5-chloropyridin-2-yl)-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperazine
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(5-methylfuran-2-yl)methyl]pyrimidin-2-amine
5-[(3S,4R)-3-carboxy-4-(3-fluorophenyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenol
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-4-ethyl-1,4-diazepan-5-one
2-(3-fluoro-4-hydroxyphenyl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
5-oxo-1-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
N-(2-methoxyethyl)-7-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide