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N-({8-[(4-methoxynaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-3-carboxamide
2-[3-(2-methylphenyl)piperidine-1-carbonyl]benzonitrile
2-{5-[1-(thiophene-3-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[2-hydroxy-3-(4-methylphenoxy)propyl]urea
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-(4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenyl)imidazolidin-2-one
3-phenyl-8-(3-propyl-1H-pyrazole-4-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
1-{[4-(2-methylpropyl)phenyl]methyl}-N-(oxan-4-yl)piperidin-3-amine
(2R,6S)-2,6-dimethyl-4-{2-[1-(2-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}morpholine
1-(2-fluoro-4-methoxyphenyl)-2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[1-(3,5-difluorophenyl)cyclopropyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
6-methyl-2-{[3-(morpholine-4-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
8-{2-[(4-methylphenyl)methyl]benzoyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-methoxy-N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-(quinoxaline-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-[(3-{[1-(3-chloro-2-methylbenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N4-ethyl-N2-methyl-N2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-2,4-diamine
(3aS,6aR)-3-cyclopentyl-5-(pyrazin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(carbamoylmethyl)-N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
(4aS,7aR)-1-(cyclopropanesulfonyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-1-methylpiperazine-2-carboxylic acid
5-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]ethyl}-2-methoxyphenol
4-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-[1-(1-benzylpiperidin-4-yl)azetidin-3-yl]pyridine
N-(2-cyclopropylphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(4aS,8aS)-2-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-decahydro-2,7-naphthyridin-4a-ol
1-(4-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}piperidin-1-yl)ethan-1-one
(2S,4R)-4-amino-N-(propan-2-yl)-1-(pyridine-4-carbonyl)pyrrolidine-2-carboxamide
(3S,4S)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
methyl 5-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-2-(phenylamino)-N-(quinoxalin-2-ylmethyl)pyrimidine-5-carboxamide
1-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-(pyridin-3-yl)benzamide
(2R,6S)-4-(2-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)-2,6-dimethylmorpholine
3-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(pyridin-3-yl)piperidin-4-ol
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-amine
(1S,2S)-1-phenyl-2-[(pyrimidin-4-yl)amino]propane-1,3-diol
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetamide
2-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)ethan-1-ol
5-amino-2-(2-methoxyphenyl)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-(3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methoxypyrazine
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carboxamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(4-aminopyrimidin-2-yl)-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-6-ol
3-[(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)oxy]pyridine