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8-[(3-hydroxyphenyl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3,3-diphenyl-1-(pyrrolidine-1-sulfonyl)piperidine
ethyl 1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
2-{5-[4-(dimethylamino)phenyl]-1H-indazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
3,5-difluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(1H-pyrazol-3-yl)phenyl]methyl})amine
N-(3-chloro-4-fluorophenyl)-N'-[2-(pyridin-4-yl)ethyl]propanediamide
(isoquinolin-5-ylmethyl)(2-methoxyethyl)(thiophen-2-ylmethyl)amine
N-{2-[2-(cyclohex-1-en-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
4-[2-(2-hydroxyphenyl)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1,2-dimethyl-1H-imidazole-4-sulfonamide
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3,6-tetrahydropyridine
2-methoxy-4-[3-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]quinoline
2-(5-acetylthiophen-3-yl)-1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
4-(dimethyl-1,2-oxazol-4-yl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-aminoethyl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1-ethyl-1,2-dihydropyridin-2-one
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-2-propyl-2,5-dihydro-1H-pyrrole-1-carboxamide
6-(4-fluorophenyl)-N-[1-(pyridin-4-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-(piperidin-3-yl)benzamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1-ethylpyrrolidine-3-carboxamide
3-butyl-1-methyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
5-(4,4-difluoropiperidine-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
(2S)-2-amino-N-(2-methylpropyl)-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
N-(2-fluorophenyl)-3-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)propanamide
1-[(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)methyl]-1H-pyrazole
[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
(4-{2-[(dimethylamino)methyl]phenoxy}phenyl)methanol
N-ethyl-2-(phenylformamido)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-amino-3-ethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetamide
(2E)-3-(3,4-dimethoxyphenyl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
3-(carbamoylmethoxy)-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)benzamide
4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(1-methylpiperidin-4-yl)amino]pyridine-3-carboxamide
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N-methyl-N-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
3-methyl-6-(5-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazol-3-yl)pyridazine
N-(4-acetylphenyl)-2-(3-methoxypropyl)piperidine-1-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-{[1-(propan-2-yl)piperidin-4-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyloxane-4-carboxamide
6-(4-fluorophenyl)-N-(2,2,2-trifluoroethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-cyclopropyl-N-[(2-methoxynaphthalen-1-yl)methyl]-6-oxopiperidine-3-carboxamide
N-benzyl-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-sulfonamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(piperazin-1-yl)pyridine-3-carboxamide
(2S)-2-amino-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pentan-1-one
[1-(3-chloro-2-fluorobenzoyl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
3-methyl-5-(5-methyl-1H-indol-3-yl)pyridin-2-amine
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropane-1-carboxamide