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N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)but-3-enamide
4-cyclobutyl-6-methyl-N-(oxolan-3-yl)pyrimidin-2-amine
methyl 3-cyclohexaneamido-5-({[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoate
6-[methyl(oxolan-3-yl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
dimethyl({5-[(5-phenylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
N-(2-chlorophenyl)-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
1-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}piperidin-2-one
{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}(propan-2-yl)amine
5-benzyl-5-{1-[(4-oxo-4H-chromen-3-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-ethyl-N-(2-hydroxyethyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
methyl 5-({[4-(methoxycarbonyl)phenyl]methyl}amino)-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,3-dimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]furan-2-carboxamide
[1-(2-methylquinolin-4-yl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
2-methoxy-N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
2-(4-{2-[(prop-2-en-1-yl)amino]benzoyl}morpholin-3-yl)acetic acid
[1-(3-chloro-4-fluorobenzoyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
[(1-{1-[(8-chloroquinolin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
3-[3-({[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]carbamoyl}amino)phenyl]-N-methylpropanamide
2-{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
3-methyl-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
(1S,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
3-methyl-1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)-3-(thian-4-yl)urea
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
1-ethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
2-(cyclopent-2-en-1-yl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
3,4,7-trimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-indole-2-carboxamide
2-(1H-pyrazol-1-ylmethyl)-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1,4-oxazepane
2-methoxy-1-{4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
1-({3-[(dimethylamino)methyl]phenyl}methyl)-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(1H-imidazol-1-yl)butan-1-one
2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-1,3-thiazole-4-carboxamide
1-(2-cyclohexylacetyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-cyclopropyl-4-[(diethylamino)methyl]-5-ethyl-N-(1,3-thiazol-5-ylmethyl)furan-2-carboxamide
(2R,3S,6R)-5-(furan-2-carbonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3-[(pyridin-3-ylmethyl)amino]benzamide
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
2-(3,4-dichlorophenyl)-4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]morpholine
N-[(1R,3R)-3-aminocyclopentyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-(3-chloro-4-propanamidophenyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
N-[2-(ethylsulfanyl)ethyl]-4-[(oxolan-3-yl)sulfamoyl]benzamide