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(3-ethyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-3-yl)methanol
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]methanol
1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[2-(pyridin-4-yl)ethyl]piperazine
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-N'-(2-methylphenyl)propanediamide
3-cyclopropyl-N-[2-(1H-indol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
6-methyl-4-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(3aR,7aS)-N-(5-fluoropyridin-3-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
ethyl({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
9-(5-acetylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclohexyl-6-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1,3-benzoxazole
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
2-(4-{[(3R)-3-aminopyrrolidin-1-yl]methyl}phenyl)-6-[(3-fluorophenyl)methyl]-3,4-dihydropyrimidin-4-one
5-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
3-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
(3aS,6aS)-5-(3-chloropyridin-2-yl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-[(5-methylfuran-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-phenylmethanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
4-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
N-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)-2-[(prop-2-en-1-yl)amino]benzamide
(3aR,7aS)-2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-(1-phenylethyl)-4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)benzamide
N-[(3S,4R)-1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-acetyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
2-(3,4-dichlorophenyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}morpholine
methyl 5-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-5-oxopentanoate
1-{2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-1H-1,2,3-triazole
3-[(2-methoxyethyl)sulfamoyl]-5-[4-(1H-pyrazol-1-yl)phenyl]benzoic acid
N-[(3S,4R)-1-(1,3-benzothiazol-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(4aS,7aR)-1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-ethyl-1H-pyrazol-5-yl)-4-[(3-methylpiperidin-1-yl)methyl]benzamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
ethyl 3-{[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]amino}propanoate
3-[5-(pent-2-yn-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(2-phenyl-1,3-thiazol-4-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]acetamide
3-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
(1S,5R)-6-{[2-(difluoromethoxy)phenyl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
4-amino-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
ethyl 4-[(6-cyanopyridin-3-yl)carbamoyl]piperazine-1-carboxylate
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-propylpyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N5-cyclopropyl-N6-[2-(pyridin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one