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[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(4-ethoxy-3-methylphenyl)butanamide
N-(2-fluoro-4-methylphenyl)-2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]acetamide
4-(3-chloro-5-fluorobenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-[4-(methylsulfanyl)benzoyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
4-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
(3S,4S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
5-methoxy-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
4-(2H-1,3-benzodioxol-5-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
3-(cyclopropylmethyl)-5-(2-fluoro-6-methoxyphenoxymethyl)-1,2,4-oxadiazole
4-[({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-6,7-dimethyl-2H-chromen-2-one
5,6-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)pyridine-3-carboxamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]-2-(pyridin-3-yl)ethan-1-ol
6-(4-ethylphenyl)-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-methyl-6-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indole
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2,4-difluorophenyl)propan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N,4-diethyl-5-methylthiophene-3-carboxamide
3-butyl-4-ethyl-1-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-methoxyphenyl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-3-carboxamide
1-methyl-6-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-1H-indole
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-(2,3-dihydro-1H-isoindol-2-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(3aR,6aR)-2-(2-cyclopentylacetyl)-5-(1H-imidazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(5-chlorothiophen-2-yl)-1-(2-methanesulfonylethyl)-1H-imidazole
6-(4-methoxy-2-methylphenyl)-N-methylpyridine-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3,5-dichlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-2-{3-[(2-fluorophenyl)formamido]propanamido}propanamide
5-(2,2-dimethylpropyl)-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(furan-2-ylmethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-(2-methylphenyl)-3-(1-{1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
4-ethyl-1-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxan-4-amine
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-cyclopropyl-N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]pyrimidine-5-carboxamide
2-methoxy-N-({5-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-{1-[(5-chloro-2-fluorophenyl)methyl]piperidin-3-yl}propan-1-ol
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
(4aR,8aR)-7-(2,1,3-benzoxadiazol-4-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
7-methyl-2-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[4-(1H-indazole-3-carbonyl)morpholin-3-yl]acetamide
(2R,4S)-4-hydroxy-1-[2-(trifluoromethyl)benzoyl]piperidine-2-carboxylic acid
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5,6-dimethyl-2-oxo-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,2-dihydropyridine-3-carboxamide
3-butanamido-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]benzamide