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7-(propan-2-yl)-2-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(2-{6-azaspiro[2.5]octan-1-ylformamido}ethyl)-2-chlorobenzamide
2-cyclopropyl-5-{4-[(2-fluorophenyl)methyl]piperazine-1-carbonyl}pyrimidin-4-ol
N-propyl-3-({5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}sulfamoyl)benzamide
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(ethoxycarbonyl)piperazin-1-yl]acetic acid
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}acetic acid
N-(furan-2-ylmethyl)-4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
ethyl 1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-ethyl-2-(3-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
4-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(8R,9aS)-2-[2-(cyclohex-1-en-1-yl)ethyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
[(2S)-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(1-methyl-5-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
5-(4-fluorophenyl)-2-methyl-4-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}pyrimidine
(3S)-3-{4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}azepan-2-one
1-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[benzyl(methyl)amino]-3-{5-[(diethylamino)methyl]-2-methoxyphenoxy}propan-2-ol
5-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(2S,4R)-1-methyl-4-({1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)pyrrolidin-2-yl]methanol
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-3-yl)pyrimidin-2-amine
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})(quinolin-5-ylmethyl)amine
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-propanoylpiperidine-3-carboxamide
2-(pyrrolidin-3-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)benzamide
1,3-dimethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-(2-{2-amino-4-[(2-methylprop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)pyrrolidin-2-one
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}-4-methoxyphenol
N-[(3R,4S)-1-(2-ethoxyacetyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]methanesulfonamide
12-(azepane-1-carbonyl)-5-chloro-9-(2-fluorophenyl)-15-methyl-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N,5-dimethyl-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-{2-[(4-oxopiperidin-1-yl)methyl]phenyl}pyridine-3-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(pyrimidin-2-ylmethyl)piperidin-4-ol
6-[(2,3-dihydroxypropyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-6-(5-methylthiophen-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}pyridine-3-carboxamide
(1S,5R)-6-(2,6-dimethylbenzoyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-methoxypropanamide
4-(2-phenylethyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N,1-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(morpholin-4-yl)benzamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(methylamino)pyridine-4-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
2-({[(3R,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol