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N-methyl-3-(2-methylphenyl)-3-phenyl-N-(pyrazin-2-ylmethyl)propanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
(3R,4S)-1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-4-propylpyrrolidin-3-amine
N-(3,4-difluorophenyl)-1-(6-methylquinoline-4-carbonyl)piperidin-3-amine
8-(2-hydroxy-4-methylbenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
(1S,5R)-3-[(5-ethylpyridin-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-benzyl-1-(3-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
methyl (2S)-1-[2-(4-{4-[(thiophen-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
1-(5-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
3,3-dimethyl-1-[(3S,4R)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
{2-[(1H-imidazol-2-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl}dimethylamine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-[2-(4-fluorophenyl)ethyl]-2-{[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]amino}acetamide
N-[5-(3-benzoylpiperidine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl]acetamide
(1R,5R)-3-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
(1R,7S)-3-(2,2-dimethylpropyl)-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}benzamide
1-(4-butylphenyl)-3-ethyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
4-amino-2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine-5-carbonitrile
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3,4,5-trimethoxybenzamide
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenol
4-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-[1-(furan-3-carbonyl)pyrrolidin-2-yl]-N-(1-methyl-1H-1,2,4-triazol-3-yl)thiophene-2-carboxamide
1-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol
4,6-dimethyl-2-oxo-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
2-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(furan-2-yl)pyrimidine
[1-(3-fluoropyridin-2-yl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
6-{1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
N-({5-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl]methanol
5-chloro-2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-methyl-1H-indole
4-methoxy-N-methyl-3-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-(3-{2-[(2,2-dimethylpyrrolidin-1-yl)methyl]-4-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
N,1,3-trimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-chloro-2-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-[4-(methylsulfanyl)phenyl]-1-(oxan-3-ylmethyl)-1H-imidazole
N-cyclohexyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(oxan-3-yl)sulfamoyl]benzamide
N-ethyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
5-(oxolane-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(4-methoxybenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
5-ethyl-1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1,3-dimethylpiperazin-2-one
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide
3-{2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione