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3-{4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
1-(2,6-dimethoxypyridine-3-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-[(2S)-2,3-dihydroxypropyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
ethyl 4-(2-methyl-4-oxo-1,4-dihydroquinoline-8-carbonyl)piperazine-1-carboxylate
(3aS,6aS)-2-(2-methoxyacetyl)-5-[(3,4,5-trifluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)pyridine-3-carboxamide
4-(3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}propoxy)benzamide
2-[(prop-2-en-1-yl)amino]-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
{2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}urea
(3E)-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}pent-3-enamide
2-[4-(dimethylamino)phenyl]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
1-(6-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}quinolin-2-yl)piperidin-3-ol
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-(pyrrolidin-1-ylmethyl)-1,3-oxazole
dimethyl[(4-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-oxazepan-6-yl)methyl]amine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(3-methylpyridin-2-yl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-[2-(dimethylamino)acetyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
N-benzyl-N-methyl-3-{1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}propanamide
N-[2-(dimethylamino)ethyl]-5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3R,4R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-3,4-dimethylpyrrolidin-3-ol
1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]piperidin-4-ol
(1s,4s)-4-hydroxy-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]cyclohexane-1-carboxamide
4-[2-amino-3-cyano-6-(4-hydroxyphenyl)pyridin-4-yl]benzamide
[1-(3,6-dimethylpyrazin-2-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
6-fluoro-2-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{[6-(methoxymethyl)pyrimidin-4-yl]amino}-2-(thiophen-3-ylmethyl)propan-1-ol
2-[3-(dimethylamino)pyrazin-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(furan-2-yl)-2-[5-methyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-phenyl-1,4-diazepane
2-[(4-chlorophenyl)methyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,3-benzoxazole
4-[(6-methylpyridin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
4-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2-(trifluoromethyl)morpholine
1-{2-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
4-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]benzonitrile
8-[4-(difluoromethoxy)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-amino-4-chloro-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-{1-[4-(1,3-oxazol-5-yl)benzenesulfonyl]pyrrolidin-2-yl}pyridine
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4-(trifluoromethyl)pyrimidin-2-amine
7-chloro-3-({[phenyl(pyridin-4-yl)methyl]amino}methyl)-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
N-(2-methanesulfonylethyl)-2-(naphthalen-2-yloxy)propanamide
4-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine
1-{[4-(methylsulfanyl)phenyl]methyl}-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
dimethyl(2-{[(2-methylphenyl)methyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amino}ethyl)amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
3-(2-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxyethan-1-one
4-{1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-(3-methylpyridin-2-yl)piperazine
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene