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1-(3,4-dichlorophenyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazine
6-methyl-2-oxo-5-({2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridine-3-carbonitrile
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
5-(3-acetylphenoxymethyl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-fluoro-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine
3-chloro-N-(2-methoxyethyl)-4-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
4-{[2-(1H-imidazol-4-yl)ethyl]sulfamoyl}-N-phenylbenzamide
N-cyclohexyl-N-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
N-benzyl-N-methyl-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-amine
5-(2,4-difluorophenoxymethyl)-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-3-carboxamide
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-{2-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]ethyl}-1H-pyrrole-2-carboxamide
5-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-[2-(dimethylamino)ethyl]-9-(2-ethylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
2-methyl-6-(3-phenylpiperazin-1-yl)pyrimidin-4-amine
6-{[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
1-(tert-butylcarbamoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
methyl (2R,4S)-1-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}-4-hydroxypiperidine-2-carboxylate
1-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}-2-methylpiperidine
5-(3,5,7-trimethyl-1H-indole-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
6-methyl-2-(pyridin-3-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
1-(2-ethoxyethyl)-5-(4-hydroxypiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclohexyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{3-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}-N-methylmethanesulfonamide
2-methyl-6-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-benzyl-3-(pyridin-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(2,6-difluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
4-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyridin-3-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]piperazine
3-(2-methoxyphenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
(3aS,6aR)-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-8-methoxyquinoline
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{4-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl}cyclobutanecarboxamide
methyl (2S)-2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2-phenylacetate
8-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
N-[(3-ethoxyphenyl)methyl]-N-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}cyclopropanamine
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
1-(cyclohexylmethyl)-6-oxo-N-propyl-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(4-fluorophenyl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
(3S,4S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(morpholin-4-yl)pyrrolidin-3-ol