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4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-1-phenylpiperazin-2-one
N-[4-({[(4-tert-butyl-1,3-thiazol-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
N-[2-(2-phenoxyethoxy)phenyl]piperidine-3-carboxamide
N-[4-(propan-2-yl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-amine
3-({5-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-3-yl}methyl)pyridine
3-fluoro-N-[2-(pyridin-3-yl)ethyl]pyridine-4-carboxamide
3-[4-(methylsulfanyl)benzoyl]-1-(thiophene-3-carbonyl)piperidine
2-[2-(dimethylamino)ethyl]-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[5-(1-cyclopropyl-1H-pyrrol-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-3-methyl-1H-pyrazole-4-carboxamide
ethyl 3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetamido]azepane-1-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethylbut-2-enamide
1-{1-[1-(furan-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}-4-methylpiperazine
3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazine
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-chloro-4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-6-methoxyphenol
(1S,5R)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-(2,4-dimethoxyphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
methyl 8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(benzyloxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-methyl-3-phenyl-8-(4-propylpyrimidine-5-carbonyl)-1,8-diazaspiro[4.5]decane
1-{4-[methyl(2-phenylethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-methyl-2,4-dioxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
9-(4-chloro-2-fluorobenzoyl)-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
3-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)propane-1,2-diol
2-(4-{[4-(furan-2-yl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)acetamide
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]thiophene-3-carboxamide
1-[2-(2-ethylphenoxy)ethyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-(3,4-dimethylphenyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
6-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-yl}pyrimidin-4-ol
N-(adamantan-2-ylmethyl)-6-{[methyl(2-phenylethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-1-[(3R,5S)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carbonyl]pyrrolidin-3-amine
(3R,4R)-3-cyclopropyl-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-methylpyrrolidin-3-ol
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-3-(3-methoxypropyl)piperidine
(3S,5R)-5-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(6-methylpyridin-3-yl)piperidine-3-carboxamide
(4aS,7aR)-1-[3-(1H-pyrazol-1-yl)propanoyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]ethan-1-one
7-(2,1,3-benzothiadiazole-4-sulfonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[2-(dimethylamino)-1-phenylethyl]-1-methyl-3-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4S)-4-cyclopropyl-1-[(1-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
propyl 4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
(1R,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-amino-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-6-(2-methylpropyl)pyrimidine-4-carboxamide