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2-{4-[3-(2-oxopiperidin-1-yl)propanoyl]piperazin-1-yl}benzonitrile
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-6-ethyl-2-methylquinoline-4-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methoxyhexan-1-one
2-[2-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
2-{1-methyl-5-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}cyclohexanecarboxamide
2-({[(3R,4R)-1-benzyl-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(pyridin-3-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1H-pyrazol-5-ylmethyl)acetamide
N-(3-fluorophenyl)-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(oxolan-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidin-4-ol
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}-4-phenylbenzamide
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
2-{3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}-7-methyl-1H-1,3-benzodiazole
5-ethyl-2-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-(cyclopropylmethyl)-5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-cyclopentyl-6-{imidazo[1,2-a]pyridin-3-yl}-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N4-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(1H-pyrrol-1-yl)ethan-1-one
5-(2-chlorophenyl)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]furan-2-carboxamide
5-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[(4-fluorophenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(3R,4R)-N-(2H-1,3-benzodioxol-5-yl)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(4-fluoro-3-methylbenzoyl)piperidin-3-yl]propan-1-ol
1-{2-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
2,3-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-7-carboxamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(quinoxalin-5-ylmethyl)amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylmorpholine-4-sulfonamide
(2S)-2-amino-1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-[2-(2-fluorophenoxy)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethan-1-amine
7-chloro-4-[1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxypropyl)-9-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4H-1,2,4-triazole
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
6-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
N5-cyclopentyl-N6-[(3-methyloxetan-3-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-(2-methoxyethyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
4-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[5-(3-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
5-{3-[4-(2-methylpropoxy)phenyl]-1H-pyrazol-5-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-cyclopropyl-2-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide