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N-benzyl-N-methyl-3-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N2-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
2-methyl-6-(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
3-{[1-(2,6-difluoro-3-methoxybenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
1-[(3,5-dimethylphenyl)methyl]-4-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]piperazin-2-one
2-(cyclohex-1-en-1-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]acetamide
4-methyl-6-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3-benzothiazol-2-amine
1-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-indole-3-carboxamide
[(3R,4R)-1-(2-ethylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[(4-chlorophenyl)methyl]-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
(1S,4S)-2-{4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carbonyl}-2-azabicyclo[2.2.1]heptane
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(thiophen-2-yl)ethyl]amine
3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-1-{4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
3-(methylsulfanyl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1,2-dimethyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
(3-{2-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(carbamoylmethyl)-N-[1-(6-methylpyridin-2-yl)ethyl]piperidine-4-carboxamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1S,2R)-1-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-2,3-dihydro-1H-inden-2-ol
5-methyl-2-(5-methylfuran-2-yl)-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
2-methyl-5-(3-{[(3,3,5,5-tetramethylcyclohexyl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-methylthian-4-amine
(4-{[1-(furan-3-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-[(3-cyclopropyl-1H-1,2,4-triazol-1-yl)methyl]-3-(diphenylmethyl)-1,2,4-oxadiazole
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3,5-dimethyl-1H-indole-2-carboxamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-2-yl)propyl]acetamide
propan-2-yl 4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(trifluoromethyl)benzene-1-sulfonamide
N-cyclopropyl-1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}piperidine-3-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-4-phenylpiperidine-4-carbonitrile
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-tert-butyl-3-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-pyrazole
(3R,9aR)-8-(naphthalene-2-sulfonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethan-1-one
1-[(2,5-dimethylphenyl)methyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
7-amino-4-(2,4-dimethoxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
8-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-{4-[3-(1-methoxyethyl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
2-methoxy-4-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
4-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}-1,4-diazepan-2-one
1-phenyl-N-[(1S,2R)-2-{[1-(propan-2-yl)piperidin-4-yl]amino}cyclobutyl]methanesulfonamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-(4-ethylpiperazin-1-yl)-3-[4-({[2-(3-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
benzyl({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine