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2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
2-[4-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N6-cyclopropyl-N5-methyl-N5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(dimethyl-1,2-oxazol-4-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propane-1,3-diol
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
5-(3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)imidazolidine-2,4-dione
1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-6-(5-methyl-1H-pyrazole-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
1-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
4-(4-methyl-1H-pyrazol-1-yl)-6-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidine
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-(2-hydroxyethyl)-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-(propan-2-yl)pyrimidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-(cyclopropylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-N-(4-methoxy-2-methylphenyl)piperidine-1-carboxamide
(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
(1S,5R)-3-{[3-(2-methylphenyl)phenyl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
3-[methyl({[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}acetamide
2-(methylsulfanyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
2-(3-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-ethylbenzamide
1-[4-(4-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
2-[3-(2-methyl-1-benzothiophen-3-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
1-[(4-acetylmorpholin-2-yl)methyl]-3-[2-(4-methoxyphenyl)phenyl]urea
1-methyl-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
2-amino-6-(3,4-difluorophenyl)-4-(1-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
1-[(2,5-dimethoxyphenyl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
N-(1-hydroxybutan-2-yl)-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
6-[(diethylamino)methyl]-N-(quinolin-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(2-methoxyethyl)-1-(pyrimidin-2-ylmethyl)piperidine-3-carboxylic acid
8-cyclopropanecarbonyl-2-(furan-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)(oxan-2-ylmethyl)amine
N-[2-(1H-imidazol-4-yl)ethyl]-2-(4-{pyrazolo[1,5-a]pyridine-3-carbonyl}morpholin-3-yl)acetamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]urea
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(propan-2-yl)pyrimidine
1-[(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3aR,6aR)-2-acetyl-N-[3-(pyridin-3-yloxy)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1H-pyrazole-5-carboxamide
1-[2-(2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]piperidine
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
methyl 3-benzamido-5-[(4-methylpentan-2-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate