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{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
1-(2-methoxyphenyl)-4-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
N-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl)pyridine-4-carboxamide
N-[(2S)-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1-oxopropan-2-yl]acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
N,8-dimethyl-3-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(3-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(oxan-4-yl)piperidin-4-amine
4-ethyl-1-methyl-3-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
3-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]azetidin-3-yl}pyridine
1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3,4,5-trimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-[3-(3,4-difluorophenyl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-[1-(2-ethylpyridine-4-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
2-cyclopropyl-8-[2-(4-methoxyphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
(2S)-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxopyrrolidine-2-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-(1,4-dioxan-2-ylmethyl)-6-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-phenyl-7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-(methoxymethyl)-N-{[3-(trifluoromethyl)phenyl]methyl}thiophene-2-carboxamide
4-methyl-6-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}pyrimidin-2-amine
3-[({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-N,N-dimethylbenzamide
8-fluoro-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}quinoline-2-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
ethyl 1-[3-({[(1-hydroxycyclohexyl)methyl]amino}methyl)-5,8-dimethoxyquinolin-2-yl]piperidine-4-carboxylate
N-(5-methanesulfonamido-2-methylphenyl)-2-phenylpyrrolidine-1-carboxamide
4-[2-(methylamino)pyridine-3-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-methoxyphenol
4-[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridine
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(3-benzyl-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)methanol
2-(3-methoxyphenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
1-methyl-5-(2-methyl-4-phenylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{2-[2-(2-phenyl-1,3-thiazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
N-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-sulfonamide
3-[5-(2,3-dichlorophenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-methyl-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1H-pyrazole-5-carboxamide
2-cyclopropyl-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 4-{4-[1-(6-fluoro-4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperazin-1-yl}benzoate
1-{1-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]propan-2-yl}-1H-1,2,4-triazole
4-(2,3-dihydro-1-benzofuran-7-yl)-7H-pyrrolo[2,3-d]pyrimidine
4-chloro-2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
4-[(3-chlorophenyl)methyl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
5-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
1-methyl-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one