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N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N,N-dimethylpropanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
3-benzyl-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
2-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)pyridine-4-carboxamide
3-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-cyclopentyl-5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidin-2-one
4-[(3-chlorophenyl)methyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
N-butyl-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(3-methylthiophene-2-carbonyl)piperidin-3-ol
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-(1-methylpiperidin-4-yl)acetamide
1-[(4aR,8aR)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(3-methoxyphenyl)ethan-1-one
6-(3-fluoro-4-methoxyphenyl)-N-(pyrrolidin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
2-(2-methoxyethyl)-8-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
5-cyclopropyl-N-(2-methoxyethyl)-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
2-{2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-6-methylpyridine
4-[2-(3-fluorophenyl)ethyl]-11-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)azetidin-3-yl]pyridine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
2-amino-3-ethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-[(prop-2-en-1-yl)amino]benzamide
4-[2-methyl-7-(oxolane-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
N3-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(morpholin-4-yl)ethan-1-one
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2,8-dimethyl-N-{3-[(pyridin-3-yl)amino]propyl}quinoline-4-carboxamide
2-[4-(benzyloxy)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
6-(1-ethyl-3-methylpiperidine-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-{2-[1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
6-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
8-{2-[4-(dimethylamino)phenyl]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2,7-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
2-cyclopropyl-3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
2-cyclopentyl-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methoxy-4-phenylpiperidine
{2-[(2,1,3-benzoxadiazol-4-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
2-(2-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-methyl-N-(pyridin-4-ylmethyl)propanamide
3-(3-{[2-(aminomethyl)morpholin-4-yl]methyl}-1H-indol-1-yl)propanamide
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
4-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-1-(4-methylphenyl)piperazin-2-one
6-cyclopentyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine