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[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N4-methyl-N2-[2-(4-methylbenzenesulfonyl)ethyl]pyrimidine-2,4-diamine
4-(piperidin-1-ylmethyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
N4-(2-methoxyethyl)-N1,N1-dimethyl-N4-(pyridin-4-ylmethyl)piperidine-1,4-dicarboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
N,N-dimethyl-3-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyrazin-2-amine
1-[(4-fluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepane
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
(4aR,7aS)-1-(2-{methyl[2-(1H-pyrazol-1-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,3-dihydro-1H-inden-2-yl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]thiolan-3-amine
2-({[1-(3-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
methyl (2S,4S)-4-(2,3-dimethyl-1H-indole-5-amido)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
3-(4-hydroxyphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
3-(1H-imidazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]butan-1-one
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-phenyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1,1-bis(furan-2-ylmethyl)urea
4-{4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
2-methoxy-N-{3-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamido]phenyl}benzamide
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[3-(1H-pyrazol-4-yl)phenyl]methyl}amine
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-tert-butyl-2-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-[2-(benzyloxy)ethyl]thieno[2,3-d]pyrimidine
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[2-(2-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-3-hydroxypyridine-4-carboxamide
5-{5-[5-(morpholin-4-ylmethyl)furan-3-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
4-[2-(2-chloro-4-methylphenoxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[(2S,4R)-4-(dimethylamino)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl]methanol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]methanol
4-(1H-imidazol-2-yl)-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidine
methyl[1-(pyrazin-2-yl)propan-2-yl]{[3-(trifluoromethyl)phenyl]methyl}amine
(1S,6R)-3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(2-{[(adamantan-1-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-(5-fluoro-2-methylphenyl)-2-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}acetamide
1-{2-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}-3,3-dimethylurea
3-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-3-enamide
4-[5-(4,6-dimethylpyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
2-ethoxy-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-4-(trifluoromethyl)benzamide
N,1-dimethyl-N-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
8-[(2R)-2-aminopropanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-methoxy-N-(2-methoxyethyl)benzamide
2-(methoxymethyl)-5-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
2-{1-cyclopentyl-4-[(2-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol