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2-(3-hydroxypropyl)-8-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-3-cyclopropyl-4-methyl-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-ol
5-(3-acetylphenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
dimethyl({3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)amine
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-[3-(propan-2-yl)-5-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxymethyl]-1H-1,2,4-triazol-1-yl]pyridine
2-{5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}pyridine
2-(2-phenyl-1H-imidazol-1-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-(cyclopropylmethyl)-4-(1H-imidazol-4-ylmethyl)-2-(propan-2-yl)-1,4-diazepane
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}benzene-1,3-diol
1-cyclobutanecarbonyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidine
5-{[2-(1H-pyrazol-1-yl)butanamido]methyl}thiophene-2-carboxylic acid
3-hydroxy-3-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1-(2-methoxyethyl)piperidin-2-one
2-[2-(3-ethylpiperazin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
2,4-dimethyl-N-{4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]phenyl}benzamide
4-[5-(2,6-dimethylpyrimidin-4-yl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl]benzamide
(1S,6R)-3-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-benzyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-thiazole-4-carboxamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)propan-1-one
3-({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
2-(1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}pyrrolidin-2-yl)ethan-1-ol
6-cyclopropyl-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidin-4-amine
6-[(1r,4r)-4-hydroxycyclohexyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
{5-methyl-7-[8-(trifluoromethyl)quinolin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-(2-fluorophenyl)-3-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)propanamide
N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
1-[4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
4-[(1-butyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,2,4-triazol-3-yl)methyl]-1-methylpiperidine
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,6-difluorophenyl)methyl]pyrrolidine-2-carboxylate
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(pyrrolidine-1-sulfonyl)piperidin-4-ol
4-(1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperidin-4-yl)morpholine
[(2S,6S)-4-[(2-chloro-6-fluorophenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-propyl-5-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
3-(5-methylfuran-2-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(5S,9aS,9bS)-5-(2H-1,3-benzodioxol-4-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
2-{[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}pyrimidine
N-methyl-2-(1-{[4-(methylsulfanyl)phenyl]methyl}-3-oxopiperazin-2-yl)acetamide
2-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-N-methylpyridine-3-carboxamide
4-(4-methylphenoxy)-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
(1-{[4-(1-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-2-yl)methanol
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
7-[3-(2-ethoxyethoxy)benzoyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1,9-dimethyl-4-[2-(1H-1,2,3-triazol-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(thiophen-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[4-({[2-(cyclohex-1-en-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide