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1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-cyclopropyl-2-{[1-(1-cyclopropylpropan-2-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
1-[3-(1H-imidazol-2-yl)-7-methylimidazo[1,2-a]pyridine-2-carbonyl]azepane
2-[2-(dimethylamino)ethyl]-9-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-3-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}propanamide
N-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
2-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidine-1-carboxamide
4,6-dimethyl-2-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]quinoxaline-2-carboxamide
4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
8-(6,8-difluoro-2-methylquinolin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
[4-({1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N,1-dimethyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}piperidin-4-amine
1'-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-(4-fluorophenyl)-N-{2-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
1-methyl-N-(3-phenylpropyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2,1,3-benzoxadiazol-4-ylmethyl)({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-indol-3-yl)ethyl]acetamide
methyl 5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3,3-dimethyl-1-(2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
2-{2-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}cyclohexanecarboxamide
3-(5-fluoro-2-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
6-(4-{[2-hydroxy-3-(4-methoxyphenoxy)propyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
3-({1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}methyl)benzoic acid
N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
4-[1-(pyridin-4-ylmethyl)piperidin-3-yl]benzoic acid
1-(1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)propan-1-ol
[7-(1,5-dimethyl-1H-indazol-3-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
6-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)piperidin-2-one
N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-phenyl-1H-pyrrole-2-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
4-methyl-N-{4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]phenyl}benzamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2R,6S)-2,6-dimethyl-4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
2-(3-methoxypropanoyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{[1-benzyl-5-(5-ethyl-1,2-oxazol-4-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
N'-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}methyl)ethanediamide
(4aS,7aR)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}propanamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-2-one
methyl (2S)-2-{[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}-2-phenylacetate
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(3S,4R)-4-(3-fluorophenyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
(2R,6S)-2,6-dimethyl-4-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine