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1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}adamantan-2-amine
4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-N,N-dimethylbenzamide
2-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
5-{[2-(dimethylamino)ethyl](oxolan-2-ylmethyl)carbamoyl}-1H-imidazole-4-carboxylic acid
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-3-yl)propan-1-one
2-{2-[(2,4-dimethyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
8-(1H-1,3-benzodiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
3-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-(4-cyclopentylpiperazin-1-yl)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)piperidine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-yl)acetamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(2-methoxyphenyl)methyl]propanamide
3-benzyl-4-[(6-methylquinolin-5-yl)methyl]piperazin-2-one
3-[(3R,4S)-1-[4-(dimethylamino)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
6-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline
N,N,4-trimethyl-5-(2-phenylazetidine-1-carbonyl)pyrimidin-2-amine
N-{[3-methyl-7-(thiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-phenyl-1H-imidazol-1-yl)acetamide
N-[(2,4-difluorophenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[2-(3-phenylpyrrolidin-1-yl)ethyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-{[(2-fluorophenyl)methyl]amino}-N-[(4-methoxyphenyl)methyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-ethyl-1-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
3-methyl-1-[1-(6-{1-oxa-7-azaspiro[3.5]nonan-7-yl}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
2-(dimethylamino)-N-[5-({[(4,6-dimethylpyrimidin-2-yl)methyl]carbamoyl}amino)-2-methylphenyl]acetamide
4-{2-[1-(furan-2-carbonyl)piperidin-2-yl]ethyl}morpholine
N-methyl-N-(2-phenylethyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
2-[(4-methylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenol
2-(2-phenylethyl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholine
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-benzyl-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-[5-(4-acetylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxyacetamide
N-(4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)cyclopropanecarboxamide
(2R)-3-(benzyloxy)-2-{[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}propan-1-ol
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
4-(3-methylpiperidin-1-yl)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]benzamide
N-ethyl-3-(4-fluorophenyl)-N-[2-(phenylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
1-benzyl-N3-[2-(2-chlorophenyl)ethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methylpropyl)-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}-N-(thiophen-3-ylmethyl)acetamide
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-[1-(4-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1,5,5-trimethylpyrrolidin-2-one
(3aS,6aR)-5-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(propane-1-sulfonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine