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4-[(2-fluoro-4-methylphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
(3ar,6ar)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl 6-({4-[methyl(phenyl)amino]phenyl}methyl)-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2,5-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-thiazole-4-carboxamide
2-[(2-methoxyethyl)(methyl)amino]-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[1-(3-methylbutanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
9-(3-fluorobenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-{2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-(5-hydroxypyrazine-2-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-8-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-acetylphenyl)-6-(1-benzothiophen-2-ylmethyl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[1-(2,6-difluoro-3-methoxybenzoyl)piperidin-4-yl]piperidin-4-ol
N-{3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]propyl}pyridin-3-amine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-(2,3-dihydro-1H-inden-1-yl)-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]-2-(1H-indol-3-yl)acetamide
7-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-methyl-6-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyridine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[7,8-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
(3S,4S)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
8-[(3-methylthiophen-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
2-[(4-methoxyphenyl)methyl]-4-[4-(quinolin-5-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)piperidin-4-ol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(4-methoxyphenyl)acetyl]piperidine-4-carboxamide
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
1-{2-[benzyl(methyl)amino]-6-phenylpyridine-3-carbonyl}piperidin-4-ol
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
6-[(2,2-dimethyloxan-4-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-(1H-pyrazol-4-yl)phenyl]urea
2-(2-chlorophenyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(N-methylmethanesulfonamido)propanamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
6-[5-(4-methoxyphenyl)furan-2-carbonyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-(methoxymethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyridine-2-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyridin-2-amine