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N-[(5-chloro-2,3-dimethoxyphenyl)methyl]-N-ethyl-2,2-dimethyloxan-4-amine
5-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
2-(3-methoxypropyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
4-{1-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrimidine
N-[(2S,4R,6S)-2-benzyl-6-(3-hydroxyphenyl)oxan-4-yl]acetamide
S-{2-[2-(dimethylamino)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-hydroxybutane-1-sulfonamido
8-cyclopropanecarbonyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,2S,9S)-N-(3-cyano-4-methoxyphenyl)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
(3aS,6aS)-2-(2-methoxyethyl)-5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-methoxyphenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyridin-2-amine
N-methyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(4-fluorophenyl)methyl]acetamide
1-[(3-fluorophenyl)methyl]-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
[3-(2-methoxyethyl)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]methanol
4-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,7aR)-1-(3-phenylpropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyano-2-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-methyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1S,5R)-3-[6-(4-methoxyphenyl)-2-oxo-1,2-dihydropyridine-3-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N,N-dimethyl-2-[(1S,5R)-6-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]thiophene-2-carboxamide
(4aS,7aR)-1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{9-[2-(3-methylphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
9-methoxy-7-(5-methylthiophen-2-yl)-4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[4-(5-methoxypyridin-3-yl)phenyl]acetamide
3-(1-methyl-1H-pyrrol-2-yl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-pyrazole-5-carboxamide
(2S)-1-(5-methyl-1,2-oxazole-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
3-[1-(2-methylpropyl)-4-phenyl-1H-imidazol-5-yl]pyridine
6-(benzyloxy)-1-cyclohexyl-4-(6-hydroxypyridine-3-carbonyl)-1,4-diazepan-2-one
3-(2,6-dimethylphenoxy)-1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidine
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(naphthalen-1-yl)ethyl]amine
1-[(3-methylpyridin-2-yl)methyl]-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazine
N-(4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)acetamide
2-cyclopropanecarbonyl-8-(4-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
5-methyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indazole
N,3,6-trimethyl-N-(quinoxalin-6-ylmethyl)-1-benzofuran-2-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
4-[2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
1-(4-methoxyphenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclopentane-1-carboxamide
N-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}methanesulfonamide
(3S,9aR)-8-(4-methylbenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}propanamide
1-(2,5-dichlorophenyl)-5-(1,4-dioxan-2-yl)-3-methyl-1H-1,2,4-triazole
2-amino-4-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1,3,6-trimethyl-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine