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2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-6-(trifluoromethyl)-1H-1,3-benzodiazole
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
1-(2-methoxybenzoyl)-4-(1H-pyrrole-3-carbonyl)piperazine
1-ethyl-9-[2-(propan-2-yl)pyrimidin-4-yl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
8-{5-[(dimethylamino)methyl]furan-2-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-indol-1-yl]-N-(propan-2-yl)acetamide
3-(cyclopropylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidine-3-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-{methyl[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-5-methylpyrazine
(1S,5R)-N-methyl-N-phenyl-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-{3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-methoxyethan-1-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-methylpyrimidine-5-carboxamide
(5-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}furan-2-yl)methanol
N-(1-hydroxybutan-2-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyrrolidin-3-yl)acetamide
3-{1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
N-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}pyrimidine-5-carboxamide
2-(adamantan-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-(2,4-difluorophenyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazole
2-(pyridin-4-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
1-methyl-4-({4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
6-methyl-4-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-[2-(4-{[3-(cyclopentyloxy)phenyl]methyl}piperazin-1-yl)ethyl]morpholine
1-[4-(furan-2-yl)benzoyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
7-(5-chloropyridin-2-yl)-4-[(2E)-3-phenylprop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3,5-dimethyl-4-(3-oxo-3,4-dihydroquinoxaline-2-amido)-1H-pyrazol-1-yl]acetic acid
2-(dimethylamino)-N-methyl-N-(2-phenyl-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl)acetamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)pyrrolidin-2-yl]methanol
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-[(2-fluorophenyl)methyl]piperidine-1-carboxamide
methyl 3-benzamido-5-{[(2,2-dimethyloxan-4-yl)formamido]methyl}benzoate
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4,6-dimethyl-2-oxo-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
3-{4-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-pyrazol-1-yl}propanamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}piperidine-1-sulfonamide
2-methyl-N-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2S,4S)-4-cyclopropaneamido-1-methyl-N-[(4-methylphenyl)methyl]pyrrolidine-2-carboxamide
(2R,3R,6R)-5-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(1H-imidazol-2-ylmethyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{4H,5H,6H,7H,8H-cyclohepta[b]thiophen-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-cyclopentyl-2-oxoacetamide
N-benzyl-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-sulfonamide
3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-[2-(3-methylphenyl)pyrimidin-5-yl]-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(2,4-difluorophenoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide