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4-[(dimethylamino)methyl]-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
N,6-dimethyl-4-oxo-N-(quinoxalin-2-ylmethyl)-4H-pyran-2-carboxamide
N-(4-methoxyphenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
2-methoxy-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-phenylacetamide
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
7-(3-chlorophenyl)-4-(2-hydroxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methylpiperidine-2-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(2,3-dihydro-1H-inden-2-yl)piperidine
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(methylamino)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-(pyridin-3-yl)-2-(pyridine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(pyridin-3-ylmethyl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepane
2-(3-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
N-[2-ethyl-4-(4-methoxy-2-methylphenyl)phenyl]acetamide
3-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
5-(2,6-difluorophenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
5-[(2S)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-(1-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(3-methylbut-2-en-1-yl)amine
3,5-dimethoxy-N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)benzamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(piperidine-1-sulfonyl)-1,4-diazepane
(3S,4S)-1-(azepane-1-sulfonyl)piperidine-3,4-diol
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
3-ethoxy-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
4-benzyl-3-ethyl-1-(2-hydroxy-5-methoxybenzoyl)-1,4-diazepan-5-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(pyridin-3-ylmethyl)amine
2-(pyridin-2-yl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(4-methylphenyl)sulfanyl]piperidine
2-methyl-6-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}pyridine
N-[4-(4-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]thiomorpholine-4-carboxamide
2-(dimethylamino)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(2-methylphenyl)acetamide
[(3S,5R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-(3-chloro-4-fluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
N-[2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]-N-methylmethanesulfonamide
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
(4S,6R)-6-methyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
(butan-2-yl)[(2,4-difluoro-3-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
7-[3-amino-3-(3,4-dimethoxyphenyl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(5-amino-4-phenyl-1H-pyrazol-3-yl)formamido]-N-(2-methylphenyl)acetamide
1-(2-ethyl-6-methylphenyl)-5-oxo-N-(4H-1,2,4-triazol-4-yl)pyrrolidine-3-carboxamide
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-8-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-methoxy-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
7-cyclohexyl-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-3-yl]methanesulfonamide
1-(2,4-difluorophenyl)-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
8-(dimethyl-1,3-thiazole-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid