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2-(3-methoxypropyl)-9-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}azetidin-3-yl)pyridine
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(3-fluoro-4-hydroxyphenyl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-(adamantan-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
(3R,4R)-1-(3-methylbutyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
3-({4-[1-(furan-2-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
3-(3-methoxyphenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-4-carboxamide
7-(1H-indole-2-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(5-ethylpyridin-2-yl)methyl]piperazine
2-methyl-6-(pyridin-2-ylmethyl)-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-(2-ethoxyethyl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-propylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 5-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[(4-methoxyphenyl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
2-cyclopropanecarbonyl-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-3-(5-methylfuran-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
1-cyclopropyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrrole-2-carboxamide
3,5,7-trimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-indole-2-carboxamide
methyl (2S,4R)-4-hydroxy-1-{[3-methoxy-5-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}pyrrolidine-2-carboxylate
6-(2-hydroxyethyl)-N-(3-phenylprop-2-yn-1-yl)-N-propylpyrazolo[1,5-a]pyrimidine-2-carboxamide
5-(4-phenoxybutyl)pyridine-3-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
1-(3-chloro-4-methoxyphenyl)-N-(cyclohex-1-en-1-ylmethyl)-5-oxopyrrolidine-3-carboxamide
6-(4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl)pyrazine-2-carboxylic acid
8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(2-fluorophenyl)-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-ethyl-4-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazin-2-one
2-fluoro-N-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methanesulfonyl-2-methylpyrimidin-4-amine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
1-(cyclohexylmethyl)-5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-[(3,4-difluorophenyl)methyl]-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
6-(2-chlorophenyl)-N-(3-hydroxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-(1-benzyl-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl)ethan-1-ol
1-[3-(1H-pyrazol-1-yl)propyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
2-{[(3-methoxypropyl)amino]methyl}-4-(6-methoxypyridin-2-yl)phenol
1-cyclopentanecarbonyl-N-(2-hydroxyethyl)-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
N-[(1-ethylpyrrolidin-3-yl)methyl]-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
1-(2,5-di-tert-butylphenyl)-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]urea
(3aR,6aR)-2-(4-ethyl-5-methylpyrimidin-2-yl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(4-methoxyphenyl)phenyl]-1-(1,2,4-oxadiazol-3-ylmethyl)piperidine-3-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
3-(4-methyl-1,3-thiazol-5-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide