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(1S,5R)-6-(5-phenyl-1,2-oxazole-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-methyl-1,2-oxazol-5-yl)-N-[2-(pyridin-3-yloxy)propyl]acetamide
N-[2-(1H-indol-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-6-(propan-2-yl)pyrimidin-2-amine
(1S,5R)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(2,4-difluorobenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
2-(4-methyl-1H-imidazol-5-yl)-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-imidazole
4-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
2-cyclopentyl-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
methyl (2S)-1-{2-[4-(4-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-3-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
3-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)-N-methylpropanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
(3S)-4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
8-(2-amino-9H-purin-6-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-oxobutanamide
1'-[1-(2-hydroxyethyl)piperidine-4-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
4-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-6-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
4-{1-cyclohexyl-5-[(2S,4R)-4-hydroxypyrrolidin-2-yl]-1H-1,2,4-triazol-3-yl}benzamide
4-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-ethoxyphenol
(2R,6S)-2,6-dimethyl-N-[2-(pyridin-2-ylmethoxy)phenyl]morpholine-4-carboxamide
N-ethyl-5-[(4-hydroxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
2-oxo-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1,2-dihydroquinoline-4-carboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]urea
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-[(5-ethylpyridin-2-yl)methyl]-1-methylurea
[2-(2-methyl-1H-indol-1-yl)ethyl][1-(1H-pyrazol-1-yl)propan-2-yl]amine
4-({5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
1-[2-(2-chlorophenyl)ethyl]-2-(oxan-2-yl)-1H-imidazole
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-(pyridin-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-(quinolin-7-yl)urea
2-{1-benzyl-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-({4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}methyl)pyridin-2-amine
5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-2-(pyrrolidin-1-yl)pyrimidine
5-methyl-3-(4-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole
5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]furan-2-carboxylic acid
8-methoxy-N-[2-(3-methylphenyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N3-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-N5-[3-(pyrrolidin-1-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-N-[(5-methylfuran-2-yl)methyl]quinazolin-4-amine
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-5-[(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)methyl]furan-2-carboxamide
N-ethyl-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(morpholin-4-yl)butanamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-pentylpyrimidine