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2-oxo-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
methyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
3-methyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
N-[(4-fluorophenyl)methyl]-N-(1-phenylethyl)pyrazine-2-carboxamide
N-(6-methylpyridin-3-yl)-1-(4-phenylbutanoyl)piperazine-2-carboxamide
3-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]quinoline
S-(2-cyclobutanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-[(4-phenyloxan-4-yl)methyl]-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]urea
1-[2-(2-fluorophenyl)ethyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
8-(4,6-dimethoxypyrimidin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane
1-[(2-fluorophenyl)methyl]-N-[(5-methylthiophen-2-yl)methyl]piperidin-3-amine
1-phenyl-3-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]propan-2-ol
5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1H-1,2,4-triazol-3-amine
N-(1,4-oxazepan-6-ylmethyl)naphthalene-1-sulfonamide
ethyl 2-oxo-5-[6-oxo-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-2,3-dihydro-1H-imidazole-4-carboxylate
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
4-(pyridin-3-ylmethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
N-[2-(methylsulfanyl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
1-(2-methyl-1-benzofuran-7-yl)-3-[3-(methylsulfanyl)propyl]urea
4-[4-(2-propylpyridine-4-carbonyl)piperazin-1-yl]quinazoline
2-[4-(dimethylamino)phenyl]-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
4-(1-ethyl-1H-imidazol-2-yl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidine
5-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-({[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
2-ethyl-8-(oxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
5-(2,5-dimethoxyphenyl)pyridin-3-amine
2-(3-methylbutyl)-8-(pyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-benzamido-5-{[(5-methyl-3-phenyl-1,2-oxazol-4-yl)formamido]methyl}benzoate
4-(1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)pyrimidine
1-({[3-(4-methyl-1,3-thiazol-2-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-ethyl-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
2-amino-4-ethyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,3-thiazole-5-carboxamide
6-fluoro-2-[4-(5-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-(2,6-dimethylphenyl)-3-[2-(methylamino)acetamido]benzamide
N-[(2R,3R)-2-methoxy-1'-(thian-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
2-[(2-oxopyrrolidin-3-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-3-carbonyl)piperidine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,3-dimethoxyphenyl)methyl]methylamine
[(2S)-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]methanol
4-methyl-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
(but-2-yn-1-yl)({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})(furan-2-ylmethyl)amine
2-{[(3R,4S)-4-cyclopropyl-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
1-{1-[2-(2,4-difluorophenyl)-1H-imidazol-1-yl]propan-2-yl}-4-methylpiperazine
1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
2-(4-fluoro-3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)acetic acid