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4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-methyl-4-{4-[1-(1-methylpiperidin-4-yl)-1H-imidazol-2-yl]phenyl}but-3-yn-2-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
3-(3-phenyl-1H-pyrazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-[(5-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}furan-2-yl)methyl]-4-methylpiperidine
1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
3-[(3-methoxypiperidin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}quinoline
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
5-chloro-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-methyl-4-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}imidazolidin-2-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(pyridin-3-ylmethyl)piperidine-1-carboxamide
2-{[3-(4-methoxyphenyl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-(methoxymethyl)-1-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-N-{3-[(pyridin-3-yl)amino]propyl}azepane-2-carboxamide
(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(6-hydroxypyrimidin-4-yl)methyl]amino}acetamide
1-ethyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-(4-fluoro-2-methylphenyl)-3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}propanamide
4-{[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-methyl-1,3-thiazole
(3S,4S)-4-propyl-1-[2-(thiophen-3-yl)acetyl]pyrrolidine-3-carboxylic acid
methyl 3-(2,2-diethylcyclopropanecarbonyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3,5-dimethylphenyl)-N-(4-ethoxy-2-fluorophenyl)-3-oxopiperazine-1-carboxamide
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(furan-2-ylmethyl)-1-methyl-3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
6-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
5-methyl-5-[1-(3-methylbutyl)piperidin-4-yl]-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]acetamide
3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-indole
(4aR,7aS)-1-cyclopropanecarbonyl-4-[2-(pyridin-2-ylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-phenylethyl)-4-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]morpholine
2-(3-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
ethyl 4-[(1-methyl-1H-indazol-6-yl)carbamoyl]piperazine-1-carboxylate
5-(2,6-dimethylphenoxymethyl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1,2-oxazole-3-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(cyclohex-1-en-1-yl)ethyl]acetamide
2-(butylsulfanyl)-6-[3-(piperidin-1-yl)pyrrolidin-1-yl]pyrimidin-4-amine
1-{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]ethyl}pyrrolidin-2-one
3-(5-methylthiophen-2-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-(4H-1,2,4-triazol-4-yl)-N-(2,4,6-trimethylpyridin-3-yl)piperidine-1-carboxamide
6-(3-methylpiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-(3-ethoxy-5-fluorophenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-fluoropyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
methyl[1-(1,2-oxazol-3-yl)ethyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-amino-4-oxo-N-[(1S)-1-phenylpropyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-[2-(furan-2-yl)phenyl]-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
1-amino-N-{2-[4-(pyridin-2-ylmethyl)morpholin-2-yl]ethyl}cyclopentane-1-carboxamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole