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1-[4-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-butyl-3-{[4-(1,1-dioxo-1λ6-thiolan-3-yl)piperazin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(propan-2-yl)-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
N-[1-(benzenesulfonyl)piperidin-4-yl]-4-(1H-pyrazol-4-yl)butanamide
1-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazole
2-(4-fluorophenoxymethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1,3-oxazole-4-carboxamide
(1R,5S,8S)-8-methoxy-3-[(5-propylfuran-2-yl)methyl]-3-azabicyclo[3.2.1]octane
methyl[(3-methyl-1H-pyrazol-5-yl)methyl]{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}amine
[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
3-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-3-ol
(4aR,7aS)-1-(2-methylpropanoyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1,5-dimethyl-1H-pyrazol-4-yl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
5-(butane-1-sulfonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(3-fluorophenyl)-3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
(3S,4R)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-[2-(piperidin-2-yl)ethyl]-5-(pyridin-2-yl)phenol
6-methyl-2-{[2-oxo-2-(4-phenylazepan-1-yl)ethyl]sulfanyl}-3,4-dihydropyrimidin-4-one
4-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(3-methylpyridin-4-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
5-ethyl-6-methyl-N4-[2-(oxan-2-yl)ethyl]pyrimidine-2,4-diamine
N-methyl-2-(pyridin-3-yl)-N-[1-(pyridin-3-yl)pentyl]pyrimidine-5-carboxamide
3-(azocane-1-carbonyl)-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
1-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-benzyl-4-[1-(2-fluorophenyl)piperidin-4-yl]-1,4-diazepan-6-ol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-cyclopropylpyrimidin-4-amine
4-methoxy-2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
5-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
methyl 1-[(3R,5S)-1-cycloheptyl-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2R)-N-[(1-benzyl-4-phenylpiperidin-4-yl)methyl]pyrrolidine-2-carboxamide
4-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]butan-1-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
3-cyclopropyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-5-carboxamide
methyl(oxan-2-ylmethyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
N-[(1-methyl-1H-indol-2-yl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1,4,6-trimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(pyridin-4-ylmethyl)-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4aS,7aR)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[propyl(pyridin-3-ylmethyl)amino]methyl}phenyl)ethan-1-one
5-{2-[(dimethylamino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-N-phenylpyrimidin-2-amine
1-(1-methylpiperidin-4-yl)-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylate
2-[(6-{4-[1-(dimethylamino)ethyl]phenyl}pyridazin-3-yl)amino]ethan-1-ol
2-[3-(adamantan-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1H-imidazole
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(1H-imidazol-2-ylmethyl)-N,1-dimethylpyrrolidine-3-carboxamide
5-({4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
4-(2-hydroxypyridine-3-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-methyl-1-[4-methyl-3-(propan-2-yl)phenyl]-3-(1-methylpyrrolidin-3-yl)urea
N-(3-{4-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]piperidin-1-yl}phenyl)-4-fluorobenzene-1-sulfonamide