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N-[2-(dimethylamino)-1-phenylethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3aR,6aS)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-fluorophenyl)-N-[1-(6-methylpyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-ethyl-6-[2-(morpholin-4-ylmethyl)phenyl]pyridazin-3-amine
4-[3-(cyclopropylmethyl)-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl]-1-ethyl-1,2-dihydropyridin-2-one
ethyl({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl})[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(furan-2-ylmethyl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(8-methoxy-2H-chromen-3-yl)methyl]methylamine
3-[(3R,4S)-1-(3-acetylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-ethyl-1H-pyrazole-5-carboxamide
N-butyl-N-[(4-fluorophenyl)methyl]-2,4-dimethylpyrimidine-5-carboxamide
2-methoxy-2-phenyl-N-[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
4-(1H-imidazol-2-yl)-1-[4-(4-methylphenoxymethyl)benzoyl]piperidine
5-(2-{5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
4-cyclopentyl-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]pyrimidin-2-amine
(1R,9S)-5-amino-3-(1-benzofuran-5-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-(2,3-dichlorophenyl)-3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
{1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}methanol
1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
4-[(2-methylphenyl)methyl]-1-(thiophen-3-ylmethyl)-1,4-diazepan-5-one
3-[(3R,4S)-1-[3-(3,5-dimethylphenyl)propanoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-(1,4-dioxan-2-ylmethyl)-6-(methoxymethyl)-N-methylpyrimidin-4-amine
2-(3-methoxyphenyl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
N-methyl-1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
[2-(dimethyl-1,2-oxazol-4-yl)ethyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-cyclopentyl-2-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)propanamide
1-[(3-fluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-fluoro-N,3-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-indole-2-carboxamide
methyl 1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
2-(pyridin-2-ylmethyl)-9-[3-(pyridin-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
N,N-diethyl-1-[(1s,4s)-4-(2-methylpropanamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
2-(1H-1,3-benzodiazol-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(3-hydroxybutyl)-1,2-oxazole-3-carboxamide
3-(azocan-1-yl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
2-methoxy-6-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-2-(naphthalen-2-yloxy)propanamide
4-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 4-{[1-(propan-2-yl)-1H-pyrazol-5-yl]carbamoyl}piperazine-1-carboxylate
5-phenyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(7-fluoro-1H-indol-1-yl)acetamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-imidazol-1-yl)propyl]amine
(4aS,8aR)-6-[2-(3-hydroxyphenyl)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
4-methoxy-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]piperidin-2-one