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4-phenyl-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-ol
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
6-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methoxy)-1,2-benzoxazole
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methyl-2-(2-methylphenoxy)butan-1-one
7-(5-methylthiophen-2-yl)-4-(9H-purin-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(thiophen-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,2,3,6-tetrahydropyridine
N-benzyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
2-(2-hydroxypropanoyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-4,6-dimethylpyridine-3-carboxamide
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[2-(thiophen-2-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-3-carboxylic acid
8-(2,4-dimethylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-4-(4-methylphenyl)-N-[2-(oxan-4-yl)ethyl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-5,6,7,8-tetrahydroquinoline-3-carboxamide
5-({[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}methyl)thiophene-2-carboxylic acid
2-butyl-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-({[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)-4-methylphenyl]propanamide
(3R,4R)-3-cyclopropyl-1-[4-(hydroxymethyl)benzoyl]-4-methylpyrrolidin-3-ol
1-{1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-yl}piperidine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(oxan-4-yl)pyrimidin-2-amine
1-ethyl-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(cyclopentylamino)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(1,3-thiazol-2-yl)piperidin-3-ol
3,5-dimethyl-1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-2-(1H-imidazol-2-yl)benzamide
1-(2-cyclohexylethyl)-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
2-methyl-5-{[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]methyl}pyrazine
N-[3-chloro-4-(2,2-dimethylpropanamido)phenyl]-5-propyl-1,2-oxazole-3-carboxamide
3-ethyl-8-{[4-(propan-2-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3,4,7-trimethyl-1H-indole-2-carboxamide
3-(3-fluorophenyl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrazole
1-methyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepane
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-oxopiperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N4-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-2-methylpyrimidine-4,6-diamine
2-[cyclopentyl(methyl)amino]-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-fluorobenzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{2-[3-cyclopentyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
2-(4-methyl-1,4-diazepan-1-yl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-{[(azepane-1-sulfonyl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(2-phenylethyl)-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
1-(3-phenylpropyl)-5-(1H-1,2,4-triazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{1-methyl-5-[(4-phenylazepan-1-yl)methyl]-1H-pyrrol-3-yl}ethan-1-one