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methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
3-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
2-ethyl-8-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(1H-indol-5-ylmethyl)morpholin-3-yl]-N-[(3-methylphenyl)methyl]acetamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}quinoline-4-carboxamide
4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-N-[(2-methylphenyl)methyl]-1,3-thiazol-2-amine
methyl 3-(2,2-dimethyloxane-4-carbonyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2,2-dimethyl-N-[1-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
(3S,4R)-1-(1H-indole-5-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
5-(3-methoxyphenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2,4-triazin-3-amine
(1S,6R)-9-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
7-(2-cyclohexylethyl)-2-[2-(pyridin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(furan-2-yl)azepane-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
1-(4-methoxybenzoyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperazine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1,4,6-trimethyl-2-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(methylsulfanyl)-3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyridine
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
6-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
2-[5-(2,6-difluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
(1S,5R)-6-[(4-ethoxyphenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 4-({6-[(diethylcarbamoyl)methoxy]-4-[(4-methoxyphenyl)methyl]-3-oxo-1,4-diazepan-1-yl}methyl)benzoate
3-chloro-4-fluoro-N-[(5-methylpyrazin-2-yl)methyl]-1-benzothiophene-2-carboxamide
N-(1-benzylcyclopropyl)-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
2-methoxy-6-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
[2-(1H-indazol-5-yl)phenyl]methanol
4-ethyl-2-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,3-thiazole-5-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(pyrrolidin-1-yl)piperidine
(2E)-3-(3,4-dimethoxyphenyl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
9-[2-(2-methoxyphenoxy)acetyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
N-[3-methyl-1-(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
2-{5-[(1S)-1-amino-5-(dimethylamino)pentyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-methyl-5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
[(3R,4R)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[4-(propan-2-yl)phenyl]methyl}piperidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
7-cyclopropanecarbonyl-N4-[(4-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-ethyl-8-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl[(4-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](quinolin-6-ylmethyl)amine
2-ethoxy-5-{2-[(1H-indol-2-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
4-[(2-methyl-1H-imidazol-1-yl)methyl]-N-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]piperidine-1-carboxamide
N-[(3R,4S)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane