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4,5-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}-2-(trifluoromethyl)pyrimidine
[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)(quinolin-2-ylmethyl)amine
6-(2,5-dimethylfuran-3-yl)-N-(2-methoxy-2-methylpropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}methanesulfonamide
3-chloro-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
{5-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
2,2-dimethylpropyl N-[(3S,5S)-1-methyl-5-{[(3S)-2-oxoazepan-3-yl]carbamoyl}pyrrolidin-3-yl]carbamate
[4-(3-phenylpropyl)-1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]methanol
8-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-5-(2-methoxyacetamido)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]propanamide
[(2-methoxyphenyl)methyl](prop-2-en-1-yl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
3-(2-ethylbutyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-7-[(2-methyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2,3-dimethoxyphenyl)methyl]-3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
5-(2-methoxyacetamido)-N-[(5-methylpyrazin-2-yl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
7-cyclopropanecarbonyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(3-fluorophenyl)-4-(3-methyl-3-phenylbutanoyl)piperazin-2-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
5-ethyl-3-{[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
ethyl 4-[(5S,9aS,9bS)-1-oxo-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
(3S,4S)-1-[4-(methylcarbamoyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-{2-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
3-({2-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenyl}-2-methylfuran-3-carboxamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylfuran-2-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxylic acid
7-[(2,3-dimethoxyphenyl)methyl]-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
6-fluoro-2-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]quinolin-4-ol
5-(2-methoxy-5-methylbenzoyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S)-2-amino-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(methylsulfanyl)butan-1-one
(2R,3R,6R)-5-(3-methyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclopentyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxamide
5-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-2-methylpyrimidine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylacetamide
N-(1,4-dimethyl-1H-pyrazol-5-yl)-3-[(4-propylpiperazin-1-yl)methyl]benzamide
5-(2,4-difluorophenoxymethyl)-N-(1,4-dioxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(4-{9-oxa-2-azaspiro[5.5]undecane-2-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
ethyl 4-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
{3-[(4-fluorophenyl)methyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl}methanol
4-[2-(3-chlorophenyl)-1H-imidazol-1-yl]benzene-1-sulfonamide
(1S,5R)-3-methyl-6-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,4S)-2-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
1-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)benzoic acid
4-(4-chlorophenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H-1,2,4-triazole
1,5-dimethyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-3-carboxamide