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1-methyl-1'-(5-propyl-1,2-oxazole-4-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{[3-(4-phenylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
methyl 4-({2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}methyl)benzoate
(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)(pyridin-2-yl)methanol
2-oxo-8-[(2E)-3-phenylprop-2-en-1-yl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(1H-pyrrol-1-yl)propyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[2-cyclopropyl-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1,2-oxazole
1-(1-benzylpyrrolidin-3-yl)-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
{5-[3-(morpholin-4-ylmethyl)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
5-amino-4-chloro-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-9H-purin-6-amine
7-[(9-ethyl-9H-carbazol-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-methyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(4aS,8aR)-6-[2-(3-chloro-4-fluorophenyl)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
5-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyridin-2-amine
N-butyl-N-[(4-fluorophenyl)methyl]-1H-pyrazole-3-carboxamide
6-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
6-(cyclobutylamino)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N-(3-fluorophenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
methyl 5-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazine
3-pentanamido-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]benzamide
N-[(3S,4R)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-methyl-5-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]quinoline
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyridin-4-ylmethyl)-decahydroisoquinoline
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
N-methyl-5-[1-(piperidin-1-yl)ethyl]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
N-(3-hydroxy-2,2-dimethylpropyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(4-methyl-5-{[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
N-cyclopropyl-3-(4-ethylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
N-({1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
N-methyl-N-(oxan-2-ylmethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-(1H-indazol-5-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(dimethylamino)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]benzamide
4-(3,5-dimethyl-1-benzofuran-2-yl)-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole
methyl 2-(cyclopropylsulfamoyl)-6-(naphthalen-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{1-[3-(1-hydroxyethyl)phenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]acetamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-methoxypropan-2-yl)acetamide
[4-(5-phenoxyfuran-2-carbonyl)-1,4-oxazepan-6-yl]methanol
4-[4-(4-benzylpiperazine-1-carbonyl)piperidin-1-yl]-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1,3-dimethyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(thiophen-2-ylmethyl)piperazine
N-[2-(1H-indol-3-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[(6-methylpyridin-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one