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1-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-(methoxymethyl)-N-(2-phenylphenyl)pyrrolidine-1-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[2-(3-methylphenoxy)phenyl]urea
(2S,4R)-N-methyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-(1,2-oxazol-3-ylmethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-(morpholin-4-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(furan-3-ylmethyl)-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
N-cyclopentyl-N-{[4-(oxolan-3-yloxy)phenyl]methyl}methanesulfonamide
N-butyl-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
N-{[3-methyl-7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
(1S,5R)-3-(3-hydroxy-4-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}oxy)pyridine
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]acetamide
1-[1-(2-fluorophenyl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
[(2S)-1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}pyrrolidin-2-yl]methanol
N-cyclobutyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
3,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(2-{[(1R,2R)-2-(diethylamino)cyclohexyl]amino}pyrimidin-4-yl)piperidin-4-ol
2-[1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)pyrrolidin-2-yl]pyridine
methyl 3-(2-cyclopentylacetamido)-6-(thiomorpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
3-[(3R,4S)-1-(3-methyl-1H-indole-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-2-yl}-N-(pyridin-2-yl)thiophene-2-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(2-methoxy-2-methylpropyl)-6-oxopiperidine-3-carboxamide
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(piperidin-1-yl)ethan-1-one
3-{5-[2-(ethylamino)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
N-({6-[4-(1H-pyrazol-1-yl)phenyl]pyridin-3-yl}methyl)acetamide
3-({3-[(4,6-dimethylpyrimidin-2-yl)amino]piperidin-1-yl}methyl)phenol
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-4-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]propan-1-one
4-(1-hydroxypropan-2-yl)-11-methyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-ethyl-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperidine
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-[(5-propyl-1H-pyrazol-3-yl)methyl]propanamide
8-({3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
2-(1-{1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(4-methylphenyl)methyl]propanamide
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1R,2R,6S,7S)-4-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(1S,5R)-3-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-methyl-1-(thian-4-yl)urea
3-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1,3-oxazolidin-2-one
methyl 6-(2,2-dimethylpropanoyl)-2-{[(3-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl[(1-methyl-1H-imidazol-2-yl)methyl][(1-phenyl-1H-pyrazol-4-yl)methyl]amine