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N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-fluoro-N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazin-2-amine
(3-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
N,N,1-triethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R)-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-phenylbutan-1-one
4-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenol
N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-methyl-6-{[1-(4-methylphenyl)propan-2-yl]amino}heptan-2-ol
2-[(4-chlorophenyl)methyl]-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-2-(2-methoxyphenyl)-1,3-thiazole
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
N-benzyl-N-cyclopentyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
1-cyclohexyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-4-carboxamide
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-2-(1H-pyrazol-1-yl)butanamide
N-[(4-hydroxyazepan-4-yl)methyl]-4-(3-methylphenoxy)benzamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-2-yl}ethan-1-ol
3-chloro-6-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
4-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
N-methyl-2-[1-(piperidin-3-yl)piperidin-4-yl]acetamide
3-{[1-(3,3,4,4,4-pentafluorobutyl)pyrrolidin-3-yl]methyl}benzamide
2-ethyl-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(2-oxopyrrolidin-1-yl)benzamide
2-{3-[({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-2-methyl-1H-indol-1-yl}acetamide
N-ethyl-5-[(3-hydroxypiperidin-1-yl)methyl]-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
methyl 4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]piperazine-1-carboxylate
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,3-benzothiazole-6-carboxamide
2-methyl-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]propanamide
N-[2-(ethanesulfonyl)ethyl]-8-fluoroquinoline-2-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
2-(5-fluoropentyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(2S,4S)-N-[(4-methylphenyl)methyl]-1-(3-phenylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(propylsulfanyl)acetamide
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyridine-4-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(morpholin-4-yl)benzamide
3-methyl-1-{1-[6-(quinolin-6-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
1-{1-[3-(dimethylamino)benzoyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-{3-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}pyrrolidin-2-one
5-methoxy-2-[3-(3-methoxypropyl)piperidine-1-carbonyl]-4H-pyran-4-one
2-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
(1S,5R)-3-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4,4,4-trifluoro-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
N,N-diethyl-1-{[4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide