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N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(quinolin-6-ylmethyl)-1H-pyrazole-4-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-3-(benzyloxy)piperidine
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(5-methylfuran-2-yl)methyl]acetamide
(1S,9R)-11-(7-methoxy-4-methylquinazolin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-[({4-[4-(2-aminoethyl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)(methyl)amino]-N-butylacetamide
3-(1H-imidazol-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
4-(5-chloro-2-methylphenyl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5,8-dichloro-3-(4-hydroxybutyl)-3,4-dihydroquinazolin-4-one
(3R,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(3-acetylphenoxymethyl)-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
3-({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
2-(2-fluorophenyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[3-(dimethylamino)-2-methylpropyl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-butyl-2-{9-oxo-4H,5H,6H,7H,8H,9H-[1,2,4]triazolo[3,2-b]quinazolin-2-yl}-N-(thiophen-3-ylmethyl)acetamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[3-(1H-1,2,3-triazol-1-yl)propyl]cyclopentane-1,3-dicarboxamide
2-(2-aminoethyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)quinazolin-4-amine
N-(3-hydroxypropyl)-N-methyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{1-[3-(2-fluorophenyl)benzoyl]pyrrolidin-3-yl}propan-2-ol
4-(1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}piperidin-4-yl)pyrimidine
1-{2-[(3-cyano-2-methoxypyridin-4-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-3-ol
2-[1-(3-methylbutyl)-4-(1-phenylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-(2-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
2-(cyclopropylmethyl)-8-(4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
ethyl 4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one
5-(3-methoxyphenyl)-4-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-2-(pyridin-4-yl)pyrimidine
methyl[(2E)-2-methylbut-2-en-1-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[(1-benzylpyrrolidin-3-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
ethyl 4-{2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetyl}piperazine-1-carboxylate
N,N-diethyl-2-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
1-[2-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
2-[(3-chlorophenyl)methyl]-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(2-chlorophenoxy)acetamide
(2S)-4-(methylsulfanyl)-2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)butan-1-ol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1,2-oxazinan-2-yl)-N-(oxolan-2-ylmethyl)propanamide
ethyl 4-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}-1H-pyrazole-3-carboxylate
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
2-[(8-chloroquinolin-2-yl)methyl]-2,8-diazaspiro[4.5]decane
1-(4-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
3-(3-hydroxypropyl)-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-methyl-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]pyridine-2-carboxamide