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3-(azepane-1-carbonyl)-1-(butan-2-yl)-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,4-dihydropyridin-4-one
3-{2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole
(furan-3-ylmethyl)(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
6-methyl-5-[5-(6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(2R,3R)-1'-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(5-propylthiophene-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
dimethyl({4-methyl-5-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(pyrimidin-2-yl)-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-1,4-diazepane
8-(1-butanoylpiperidin-4-yl)-2-ethyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N,N-dimethyl-4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
4-{5-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]furan-2-yl}-2-methylbut-3-yn-2-ol
7-methyl-2-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(propan-2-yloxy)ethyl]propanamide
7-{[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]sulfonyl}-2-oxa-7-azaspiro[4.5]decane
3-ethyl-8-(6-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
N,N-dimethyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
[1-(5-chloropyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methanol
3-{1-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}benzonitrile
4-(2,2-dimethyloxan-4-yl)-1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-1,2,3-triazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-6-oxo-N-(oxolan-2-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(4-methoxyphenyl)-N-[2-(1-methylpiperidin-3-yl)ethyl]cyclopropane-1-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-(6-cyanopyridin-3-yl)-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
N-[(3R,4R)-1-(6,8-dimethylquinolin-4-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-[ethyl(methyl)amino]-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
9-(2-hydroxyethyl)-1-methyl-4-(pyridine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,8aS)-2-(3-methoxy-5-methylthiophene-2-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(4-fluorophenyl)ethyl]-5-methoxybenzamide
3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
(3E)-N-butyl-N-[(2-methylphenyl)methyl]pent-3-enamide
6-(4-methoxyphenyl)-2-(4-{[methyl(propan-2-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(2,1,3-benzoxadiazol-5-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-benzyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
(4aS,8aS)-2-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-decahydroisoquinolin-4a-ol
6-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{1-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]piperidin-2-yl}methanol
2-(diethylamino)-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3,4,7-trimethyl-2-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-1H-indole
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-({1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-({[1-(methoxymethyl)cyclopentyl]methyl}sulfamoyl)-N-propylbenzamide
3-(1,3-benzothiazol-2-yl)-1-[4-(furan-2-carbonyl)piperazin-1-yl]propan-1-one
4-methyl-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-3-(2-oxoimidazolidin-1-yl)benzamide
1-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one