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N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
(3S)-3-ethyl-4-(4-methyl-2-phenylpyrimidine-5-carbonyl)morpholine
(2S)-2-(dimethylamino)-3-phenyl-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-[3-(1H-pyrazol-1-yl)phenyl]-5-(thiomorpholine-4-sulfonyl)benzoic acid
4-butyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(3R,5S)-5-(4,4-difluoropiperidine-1-carbonyl)pyrrolidin-3-yl]-3-methoxypropanamide
ethyl 2-(N-methyl-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)acetate
4-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl](methyl)amino}methyl)-1-methylpyrrolidin-2-one
6-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine
2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
4-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]piperazine-2-carboxylic acid
4-{4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
ethyl 1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(butan-2-yl)-6-oxo-N-(pyridin-4-ylmethyl)-1,6-dihydropyridine-2-carboxamide
3-{[4-(3-ethenylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
2-{5-[3-(azepan-1-ylmethyl)phenyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}acetic acid
3-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}benzoic acid
1-cyclopentyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-6-oxopiperidine-3-carboxamide
3-methyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
2-(3-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-amine
N4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-(thiophen-2-ylmethyl)benzamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-ol
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(2,5-dimethylphenyl)methyl]amino}-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
5-(4,6-dimethoxypyrimidin-2-yl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(pyridin-3-yl)propanamide
6-[2-(4-hydroxyphenyl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
3-amino-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2H-1,3-benzodioxole-5-carboxamide
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-4-methyl-1,2,5-oxadiazole
N-{4-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
2-(methoxymethyl)-5-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)pyrimidine
3-[4-(3-methoxypropyl)piperidin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}benzamide
1,3-dimethyl-6-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,3,5-trimethyl-N-(prop-2-en-1-yl)-1H-indole-2-carboxamide
3-[3-(1,3-benzoxazol-2-yl)phenyl]propanamide
1-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-3-methylbutan-1-ol
(2S)-2-amino-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxypropan-1-one
4-(4-methylphenoxy)-N-[(5-methylpyrazin-2-yl)methyl]piperidine-4-carboxamide
4-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(oxolan-3-yl)-5-(5-propyl-1,2-oxazol-3-yl)-1,2,4-oxadiazole
2-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-methanesulfonylethan-1-one
1-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one