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5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
3-(3,4-difluorophenyl)-5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(4-methylphenyl)acetamide
ethyl 4-benzyl-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine-4-carboxylate
7-fluoro-4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-({3-methyl-7-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
3-methoxy-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-(oxan-4-yl)-3-(4-phenoxybenzoyl)piperidine
N-[3-(1H-1,2,3-triazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(3R,4R)-3,4-dimethyl-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-2,2-dimethylthiomorpholin-3-one
2-amino-6-hydroxy-4-(4-hydroxy-2-methoxyphenyl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
2-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-2-yl}pyridine
(3S)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-N,N-dimethylazepan-3-amine
6-phenyl-N-[2-(propane-2-sulfonyl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-acetyl-N-(9H-fluoren-9-yl)-1H-pyrazole-5-carboxamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(3-fluorophenoxymethyl)piperidine
1-(2-chlorophenyl)-5-methyl-4-(6-methylpyridine-2-carbonyl)piperazin-2-one
2-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}acetamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-4-(oxolan-2-ylmethyl)piperazine
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)(2-phenylethyl)amine
N-[(2-fluorophenyl)methyl]-3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(dimethylamino)-N-ethyl-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide
1-methyl-2-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-1,3-benzodiazole
N1-(1,4-dithiepan-6-yl)-N2-(pyridin-3-yl)ethane-1,2-diamine
N-[(3R,4R)-3-hydroxy-1-[2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
4-ethyl-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-(4-methoxybenzamido)-1-methyl-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-{4-[(4-cyclopentylpiperazin-1-yl)methyl]phenoxy}-3-(dimethylamino)propan-2-ol
1-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
1-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(2-oxopiperidin-1-yl)propanamide
2-[(3-{[1-(thiophen-2-yl)propan-2-yl]carbamoyl}phenyl)amino]acetic acid
2-(4-hydroxyphenyl)-N-(propan-2-yl)pyridine-4-carboxamide
3-hydroxy-3-({[(4-methylphenyl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-cyclopentyl-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
(2S)-N-ethyl-5-oxo-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
8-(5-chloro-2-fluorobenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]azetidin-3-yl}pyridine