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5-{2-[(prop-2-en-1-yl)amino]ethyl}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-(2,3-dihydro-1H-inden-1-yl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-indole-6-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-[(3-chlorophenyl)methyl]-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
2-{[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)phenyl]amino}acetic acid
ethyl 4-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]piperidine-1-carboxylate
4-(azonan-1-yl)-N-cyclopentyl-4-oxobutanamide
6-(1-benzofuran-2-yl)-N,N-dimethylpyridine-2-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-[(1-propyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclobutylmethyl)-2-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-oxo-1-[(2-phenylphenyl)methyl]pyrrolidine-3-carboxylic acid
(1S,5R)-3-(3,5-dimethylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-2-methyl-1H-indole-3-carbonitrile
4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-2-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1-(4-methyl-2-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-5-yl)ethan-1-one
(1S,5R)-6-(2-methyl-1-benzofuran-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[benzyl(methyl)amino]-3-[4-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-methyl-1-{[3-(3-propylmorpholine-4-carbonyl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole
4-[(dimethylamino)methyl]-1-[2-(pyrrolidin-1-yl)benzoyl]azepan-4-ol
2-(morpholin-4-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-oxazepane
2-ethoxy-5-(2-methoxypyridin-3-yl)benzamide
1-{2-[1-(6-methylquinolin-4-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-(4-benzylpiperidin-1-yl)-3-[1-(3-methoxybenzoyl)piperidin-4-yl]propan-1-one
N-(4-chloro-3-methoxyphenyl)-2-{[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amino}acetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(2,1,3-benzoxadiazol-5-ylmethyl)acetamide
2-(3-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-({[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]amino}methyl)pyrrolidin-3-ol
7-methyl-2-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
5-phenyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(4-{2,8-diazaspiro[4.5]decan-2-ylmethyl}phenyl)prop-2-yn-1-ol
2-{8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)-1H-1,3-benzodiazole
N-[1-(4-methylphenyl)ethyl]-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetamide
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-3-(3-methoxypropyl)piperidine
5-methoxy-3-methyl-2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
3-(2-ethyl-1H-imidazol-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}propanamide
1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)azepane
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-(5-phenyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3-methoxybenzoyl)-4-(1H-pyrrole-3-carbonyl)piperazine
(1S,5R)-6-(5-methylpyrazine-2-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{5-[(3,4-difluorophenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
1-methyl-3-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indol-2-one