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N-ethyl-N-(2-methoxyethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(2S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(carbamoylmethyl)-N-{1-[4-(dimethylamino)phenyl]propan-2-yl}piperidine-4-carboxamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-4-methyl-1,3-oxazole-5-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(pyridin-3-ylmethyl)-3-[1-(quinoxalin-2-yl)piperidin-4-yl]propanamide
N-(1-{4-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
1,9-dimethyl-4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
(3aR,6aR)-2-(2-chlorobenzoyl)-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(furan-3-ylmethyl)-N,2,4-trimethylpyrimidine-5-carboxamide
3-(2-fluorophenoxy)-1-[(4-methoxyphenyl)methyl]azetidine
2-methoxy-5-{[methyl(quinolin-6-ylmethyl)amino]methyl}benzoic acid
1-methyl-2-(morpholin-4-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-[1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-5-yl]butanoic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidine-3-carboxylic acid
N-[2-(quinolin-8-yloxy)ethyl]pyrimidin-4-amine
N-{5-[({1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)methyl]-1,3-thiazol-2-yl}pyridin-3-amine
N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]-2-[3-(trifluoromethyl)phenyl]acetamide
2-(3-methoxypropyl)-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(pyridin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]quinoline-4-carboxamide
N-[(3-chlorophenyl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-propylacetamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
2-(3-methoxyphenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}azepane
1-(4-methoxyphenyl)-4-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperazine
1-[3-(2-methylphenyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(pyrazin-2-yl)ethyl]pyrimidin-2-amine
4-(5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl)pyridine
5-cyclopropanecarbonyl-1'-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-2-[1-({[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(2-methoxyphenyl)propan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyrimidin-4-ol
ethyl 4-[2-(5-acetylthiophen-3-yl)acetamido]piperidine-1-carboxylate
2-[2-methyl-3-({[4-(pyridin-2-yl)butyl]amino}methyl)-1H-indol-1-yl]acetamide
methyl 3-[(2E)-3-(2-chlorophenyl)prop-2-enamido]-5-{[(1-methylpiperidin-2-yl)formamido]methyl}benzoate
4-{4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperazine-2-carbonyl}morpholine
2,8-dimethyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
2-(benzyloxy)-1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
3-{[1-(4-sulfamoylbutanoyl)pyrrolidin-3-yl]methyl}benzamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}ethane-1-sulfonamide
4-ethyl-6-(1H-pyrazol-3-yl)-2-(pyrrolidin-1-yl)pyrimidine
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-2-(methylamino)benzamide
1-{4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4-oxobutyl}pyrrolidin-2-one
(2-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide