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diethyl({3-[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(3S,4S)-1-[2-oxo-2-(piperidin-1-yl)ethyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
[1-phenylmethanesulfonyl-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline
4-phenoxy-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
1-methyl-1'-(pyridine-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(4-{thieno[2,3-d]pyrimidin-4-yl}morpholine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-[5-(3-chloro-4-fluorobenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
3-{3-[({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
4-[3-(2-methoxyphenoxy)azetidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)morpholine-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
(1s,4s)-4-hydroxy-N-[1-(pyridin-3-yl)pentyl]cyclohexane-1-carboxamide
2-methyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]furan-3-carboxamide
N-[1-(3,5-difluorophenyl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(pyridin-3-yloxy)ethyl]benzamide
2-(propan-2-yl)-9-(pyridin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(5-propyl-1,2-oxazole-3-carbonyl)-6-azaspiro[2.5]octane
1-({[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}methyl)cyclohexan-1-ol
3-(3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}piperidine-1-carbonyl)pyridine
1-[3-({3-[2-(methoxymethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
1-(2,1,3-benzothiadiazol-5-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-1-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
(1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}piperidin-3-yl)methanol
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
methyl 3-(2-phenylacetamido)-5-[(1,2,5-thiadiazol-3-ylformamido)methyl]benzoate
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
3-(1H-indazol-7-yl)-1-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}urea
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2,2-dimethylbutan-1-one
2-benzyl-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N,N-bis(1,3-oxazol-4-ylmethyl)-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(4,6-dimethylpyrimidin-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2R,6R)-4-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2,7,8-trimethyl-4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]quinoline
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methylphenol
N-methyl-N-phenyl-2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]benzamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[3-(dimethylamino)propyl]-N-methyl-1,3-oxazole-4-carboxamide
1-tert-butyl-4-{[methyl(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}pyrrolidin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-methyl-9-(prop-2-en-1-yl)-4-(1,3-thiazol-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(2-chloro-4-fluorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-{4-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxymethyl}pyridine
2-(2-oxoazepan-1-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
8-[(4-fluorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea