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N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
6-(propan-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-2-(trifluoromethyl)pyrimidin-4-amine
5-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-methoxy-2-methylpropan-1-one
4-(1H-imidazol-1-ylmethyl)-1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-4-ol
3-(2-methoxyethyl)-5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1,2,4-oxadiazole
3-{2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetyl}piperidine-4-carboxamide
4-{1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}morpholine
N-{2-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-oxoethyl}acetamide
N-[5-({[(4,6-dimethylpyrimidin-2-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]-2-methoxyacetamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
3-(3-ethoxypropyl)-1-[4-(4-methoxyphenyl)phenyl]urea
(3S,9aR)-3-benzyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{6-[1-(2-ethoxyethyl)piperidin-3-yl]-2-methylpyrimidin-4-yl}morpholine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]pyrimidin-2-amine
3-[(3R,4S)-1-(3-chloro-4-methoxybenzoyl)-4-(dimethylamino)piperidin-3-yl]propanoic acid
(3S)-1-ethyl-3-methyl-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazin-2-one
7-cyclopropanecarbonyl-N-[(5-methylpyrazin-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2,5-thiadiazole
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylpentanamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
3-methyl-6-[4-(pyridin-4-yl)piperidin-1-yl]pyridazine
[9-benzyl-3-(1H-pyrrole-2-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-(4-{[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-5-methyl-1-propyl-1H-pyrazole
1-[4-(piperidine-1-carbonyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-1H-indole
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(3-methoxyphenyl)-1,3-thiazole
4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]morpholine
1-(4-fluorophenyl)-4-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-3-yl}piperazine
butyl 8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
2-{5-[3-(1H-imidazol-2-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)-N-(2-methylpropyl)acetamide
8-(1,3-benzothiazol-2-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(pyridin-4-yl)piperidine-1-carboxamide
3-({[(1-ethyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
2-methoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)acetamide
2-{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(pyridin-3-yl)acetamide
1-{[4-(dimethylamino)phenyl]methyl}-4-(2-phenoxyethyl)-1,4-diazepan-5-one
methyl 3-[1-(phenylcarbamoyl)-6-azaspiro[2.5]octane-6-carbonyl]benzoate
9-(2-ethoxyacetyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
7,7-dimethyl-2-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
2-(4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
9-{[4-(trifluoromethoxy)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane