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ethyl 4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazine-1-carboxylate
2-fluoro-6-hydroxy-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)benzamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(3-hydroxypropyl)benzamide
{3-[2-(1-{5-[(dimethylamino)methyl]pyridin-2-yl}piperidin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
3-[(4-methyl-6-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}pyrimidin-2-yl)amino]phenol
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-[(dimethylamino)methyl]furan-2-carboxamide
ethyl 3-(2-phenoxyethyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
2-methyl-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrrolidin-1-yl)propan-1-one
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4-(1,3-thiazol-2-yl)piperazine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
4-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(2-methoxyethyl)piperazine
N-[(2R,3R)-1'-(isoquinolin-5-ylmethyl)-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecane-3-carbonyl]cyclopentan-1-ol
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-(2-methanesulfonylethyl)benzamide
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(oxane-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-ethyl-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-methoxy-5-{1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-imidazol-2-yl}phenol
9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
1-(2,3-dihydro-1H-inden-4-yl)-3-(2-methoxyethyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
1-(2,2-dimethylpropanoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(piperidin-1-ylmethyl)piperidine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(4-chlorophenyl)butanamide
N-cyclopropyl-4-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
6-methyl-5-{2-[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[cyclohexyl(methyl)amino]-3-(3-{[(thiophen-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
5-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}amino)-N,N-dimethyl-1-benzothiophene-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
{5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
[1-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
[(1-cyclopentylpiperidin-4-yl)methyl][(3-fluorophenyl)methyl](pyridin-3-ylmethyl)amine
1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
2-cyclopropyl-8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-methyl-4-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-benzyl-N-(4-methoxyphenyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[(4-methoxyphenyl)methyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
8-methoxy-N-methyl-N-(quinolin-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aS,8aR)-1-butyl-6-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
[(2-{[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methyl]dimethylamine
(3S,4S)-4-cyclopropyl-1-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)pyrrolidine-3-carboxylic acid
3-(5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
(2E)-1-[(4aR,8aR)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-6-yl]-2-methylbut-2-en-1-one
N-tert-butyl-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-(2-oxoazepan-3-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(2S)-2-hydroxy-2-phenylethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide