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2-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]piperidin-1-yl}-4,6-dimethylpyrimidine
5-[(dimethylamino)methyl]-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-2-carboxamide
2-[3-(pyridin-4-yl)-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
3-methyl-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[7-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-hexyl-2-(4-methylpiperazin-1-yl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
N-(2-fluoro-5-methylphenyl)-N'-methyl-N'-[1-(pyrimidin-4-yl)ethyl]butanediamide
(2S,3S)-3-methyl-2-{[(2-methyl-5-sulfamoylphenyl)carbamoyl]amino}pentanamide
methyl 3-[(3S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
2-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetamide
2-chloro-5-acetamido-N-(oxolan-2-ylmethyl)benzamide
[(3R,4S)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,3,5-trimethyl-1H-pyrazole-4-carboxamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-[4-(2,5-dimethylthiophene-3-sulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(pyridin-3-yl)prop-2-enamide
methyl 2-{2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamido}acetate
4-[2-(benzyloxy)acetyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(cyclopropylmethyl)-N-propyl-1,3-oxazole-4-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-(3,4,5-trimethoxyphenyl)acetamide
6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-{9-[(2-methylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-{[(2R,5S)-5-(1-benzofuran-5-ylmethyl)oxolan-2-yl]methyl}-N,1-dimethylpiperidin-4-amine
N-cyclopropyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}thiophene-2-carboxamide
N,N-diethyl-1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(4-hydroxybenzoyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-chlorophenyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-phenylpropanamide
methyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5-methyl-6-(5-methylthiophen-2-yl)pyridine-3-carbonitrile
1-methyl-8-{[methyl(phenyl)carbamoyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 1-[3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
1-(2-methoxy-5-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
benzyl(methyl){[3-(4-propyl-1,4-diazepane-1-carbonyl)-1,2-oxazol-5-yl]methyl}amine
1-methanesulfonyl-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine
methyl 2-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamido]acetate
8-(5-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-chloro-4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]phenol
N-[3-(cyclohexylcarbamoyl)-2-methylphenyl]oxolane-3-carboxamide
2-(2-ethoxypyridin-3-yl)-2-(morpholin-4-yl)acetic acid
N6-cyclopropyl-N4-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N4-methylpyrimidine-2,4,6-triamine
5-{[(3-hydroxy-3-phenylpropyl)(methyl)carbamoyl]amino}-2-methoxy-N-methylbenzamide
3-(2-methylphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-ol
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[3-(furan-2-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-cyclopropanecarbonyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]pyrrolidine-2-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-5,6-dimethyl-1H-1,3-benzodiazole